Bromide

Bromide

SCHEMBL998627

Br.c1ccc(CNCc2ccccc2)cc1

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 1/20 0.61
SIGMAR1 known ✓ Q99720 3/20 0.56
MEN1 O00255 1/20 0.74
KMT2A Q03164 1/20 0.74
TDP1 Q9NUW8 1/20 0.74
MAOA P21397 1/20 0.64
MAPT P10636 3/20 0.61
GAA P10253 1/20 0.61
PKM P14618 1/20 0.58
BCHE P06276 1/20 0.58
IDO1 P14902 2/20 0.57
THRB P10828 1/20 0.57
ADH1B P00325 1/20 0.56
ADH1C P00326 1/20 0.56
ADH1A P07327 1/20 0.56
ADH7 P40394 1/20 0.56
CYP3A4 P08684 2/20 0.55
KDM4E B2RXH2 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1654 0.97 MEN1 (0.78) MEN1KMT2ATDP1MAOAMAPT
SCHEMBL5799878 0.97 MEN1 (0.78) MEN1KMT2ATDP1MAOAMAPT
Benzene SCHEMBL11697595 0.97 MEN1 (0.78) MEN1KMT2ATDP1MAOAMAPT
Fluoride SCHEMBL634375 0.94 MEN1 (0.74) MEN1KMT2ATDP1MAOAMAPT
SCHEMBL21550054 0.94 MEN1 (0.74) MEN1KMT2ATDP1MAOAMAPT
Ammonia Solution, Strong SCHEMBL2064651 0.94 MEN1 (0.74) MEN1KMT2ATDP1MAOAMAPT
SCHEMBL3990993 0.94 MEN1 (0.74) MEN1KMT2ATDP1MAOAMAPT
Hydrochloric Acid SCHEMBL1862144 0.94 MEN1 (0.74) MEN1KMT2ATDP1MAOAMAPT
Water SCHEMBL11666905 0.94 MEN1 (0.74) MEN1KMT2ATDP1MAOAMAPT
SCHEMBL30223761 0.94 MEN1 (0.74) MEN1KMT2ATDP1MAOAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119350290-A Method for preparing 1, 4-dioxane-2-ketone from ethylene carbonate 青岛科技大学 2025-01-24 CN disclosed
EP-2451792-A2 PROCESS FOR SUBSTITUTED 3-AMINO-5-OXO-4,5-DIHYDRO-[1,2,4]TRIAZINES OSI Pharmaceuticals, LLC (US) 2012-05-16 EP disclosed
CN-101560171-B Preparation method of 5- (N, N-dibenzylglycyl) salicylamide JIANDE ZISHANWAN FINE CHEMICAL CO LTD 2012-05-09 CN disclosed
US-20120108812-A1 PROCESS FOR SUBSTITUTED 3-AMINO-5-OXO-4,5-DIHYDRO-[1,2,4]TRIAZINES OSI PHARMACEUTICALS ,INC. 2012-05-03 US disclosed
WO-2011005909-A2 PROCESS FOR SUBSTITUTED 3-AMINO-5-OXO-4,5-DIHYDRO-[1,2,4]TRIAZINES OSI PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed
CN-101560171-A Method for preparing 5-(N,N-dibenzylglycyl) salicylamide JIANDE ZISHANWAN FINE CHEMICAL (CN) 2009-10-21 CN disclosed
EP-1009447-B1 HYDROXYMETHYL PHOSPHINE COMPOUNDS FOR USE AS DIAGNOSTIC AND THERAPEUTIC PHARMACEUTICALS AND METHOD OF MAKING SAME UNIV MISSOURI (US) 2005-08-10 EP disclosed
US-20030045727-A1 Process for preparing optically active secondary alcohols having nitrogenous or oxygenic functional groups ASAHI KASEI KABUSHIKI KAISHA (JP) 2003-03-06 US disclosed
EP-1254885-A1 PROCESS FOR PREPARING OPTICALLY ACTIVE SECONDARY ALCOHOLS HAVING NITROGENOUS OR OXYGENIC FUNCTIONAL GROUPS Asahi Kasei Kabushiki Kaisha (JP) 2002-11-06 EP disclosed
EP-1009447-A4 HYDROXYMETHYL PHOSPHINE COMPOUNDS FOR USE AS DIAGNOSTIC AND THERAPEUTIC PHARMACEUTICALS AND METHOD OF MAKING SAME UNIV MISSOURI (US) 2001-04-11 EP disclosed
WO-1998041242-A1 HYDROXYMETHYL PHOSPHINE COMPOUNDS FOR USE AS DIAGNOSTIC AND THERAPEUTIC PHARMACEUTICALS AND METHOD OF MAKING SAME THE CURATORS OF THE UNIVERSITY OF MISSOURI (US) 1998-09-24 WO disclosed
US-5405872-A Anti-hypertensive tetralins BURROUGHS WELLCOME CO. (US) 1995-04-11 US disclosed
EP-0549668-A1 ANTI-HYPERTENSIVE TETRALINS THE WELLCOME FOUNDATION LIMITED (GB) 1993-07-07 EP disclosed
US-5194450-A Hypotensive agents BURROUGHS WELLCOME CO. (US) 1993-03-16 US disclosed
US-5102914-A Racemic mixtures BURROUGHS WELLCOME CO. (US) 1992-04-07 US disclosed
WO-1992005143-A1 ANTI-HYPERTENSIVE TETRALINS THE WELLCOME FOUNDATION LIMITED (GB) 1992-04-02 WO disclosed
US-4336400-A BRONCHODILATOR AGENTS, CARDIOVASCULAR STIMULANTS STERLING DRUG INC. (US) 1982-06-22 US disclosed
EP-0030030-A1 Derivatives of 2-aminoethanol, processes for their preparation, pharmaceutical compositions containing such compounds and the use the latter CIBA-GEIGY AG (CH) 1981-06-10 EP disclosed
US-4138581-A BRONCHODILATOR AGENTS, ADRENERGIC STIMULANTS STERLING DRUGS INC. (US) 1979-02-06 US disclosed
US-4101579-A Phenethanolamine ethers ALLEN & HANBURYS LIMITED (GB) 1978-07-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030045727-A1 Process for preparing optically active secondary alcohols having nitrogenous or oxygenic functional groups ADH1A, ADH5, ADH1C CHRM2 110/4885SIGMAR1 42/4885MEN1 3345/4885
US-20120108812-A1 PROCESS FOR SUBSTITUTED 3-AMINO-5-OXO-4,5-DIHYDRO-[1,2,4]TRIAZINES ALKBH5, NT5C, CYP4Z1 CHRM2 2062/4885SIGMAR1 1634/4885MEN1 2700/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.