SCHEMBL9988702

SCHEMBL9988702

COc1ccc(-n2nc(CCC(=O)NCCN3CCOCC3)cc2-c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.58
KDM5B Q9UGL1 2/20 0.56
POLB P06746 2/20 0.55
RXRA P19793 1/20 0.51
RXRB P28702 1/20 0.51
RXRG P48443 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
ALOX5 P09917 1/20 0.49
RPA1 P27694 1/20 0.48
MMP2 P08253 1/20 0.47
MMP8 P22894 1/20 0.47
MMP12 P39900 1/20 0.47
MMP13 P45452 1/20 0.47
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9988404 0.95 PTGS2 (0.59) PTGS2KDM5BPOLBRXRARXRB
SCHEMBL9988387 0.88 DRD4 (0.49) PTGS2KDM5BPOLBKDM4EHSD17B10
SCHEMBL9989269 0.86 PTGS2 (0.54) PTGS2POLBRXFP1KDM4E
SCHEMBL9989347 0.85 RXRA (0.49) PTGS2RXRARXRBRXRGALOX5
SCHEMBL9988533 0.83 LMNA (0.49) PTGS2KDM5BPOLBRXRARXRB
SCHEMBL9988392 0.82 MC4R (0.57) PTGS2RXRARXRBRXRGALOX5
SCHEMBL9989304 0.81 RXRA (0.52) PTGS2POLBRXRARXRBRXRG
SCHEMBL9989355 0.81 MALT1 (0.62) PTGS2RXRARXRBRXRGKDM4E
SCHEMBL9989408 0.79 DRD4 (0.51) POLBRXRARXRBRXRGKDM4E
SCHEMBL9988308 0.78 MALT1 (0.55) PTGS2RXRARXRBRXRGALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011161615-A1 5-LIPOXYGENASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2011-12-29 WO disclosed