SCHEMBL10069618

SCHEMBL10069618

CC(C)c1c(-c2cccc3ccccc23)n(COCc2ccc(Cl)cc2F)c(=O)n(O)c1=O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 5/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
MAPK14 Q16539 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
TBXA2R P21731 2/20 0.33
PTGS1 P23219 2/20 0.33
CYP2C19 P33261 2/20 0.33
PTGER3 P43115 2/20 0.33
PTGER2 P43116 2/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
RAB9A P51151 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
HPD P32754 2/20 0.32
PTGES O14684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10069624 0.87 GHSR (0.33) PTGER1AKR1C3AKR1C2MAPK14CYP1A2
SCHEMBL10069599 0.84 PTGS2 (0.34) PTGER1AKR1C3AKR1C2PTGS1MEN1
SCHEMBL10069626 0.83 HPD (0.34) PTGER1MAPK14CYP1A2CYP2C9TBXA2R
SCHEMBL10069593 0.82 MEN1 (0.35) MAPK14MEN1KMT2AHPD
SCHEMBL10069608 0.82 HPD (0.32) MAPK14HPD
SCHEMBL10069609 0.81 LMNA (0.34) MAPK14MEN1KMT2AMAPK1HPD
SCHEMBL10069607 0.81 ADORA2A (0.35) MAPK14HPD
SCHEMBL10069594 0.71 MAPT (0.38) CYP1A2KDM4E
SCHEMBL10069596 0.70 MAPT (0.36) MAPK14CYP1A2CYP2C9MEN1KMT2A
SCHEMBL10069590 0.67 ALDH1A1 (0.39) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed