SCHEMBL10075868

SCHEMBL10075868

Cc1ccc(C(=O)c2ccc(I)cc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.76
LMNA P02545 2/20 0.76
SRD5A2 P31213 2/20 0.64
CES2 O00748 2/20 0.54
CES1 P23141 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.52
TPMT P51580 1/20 0.52
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
AKR1C3 P42330 1/20 0.48
HTT P42858 3/20 0.48
PKM P14618 2/20 0.48
ATM Q13315 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
HPGD P15428 1/20 0.48
NLRP1 Q9C000 1/20 0.48
GAA P10253 1/20 0.48
MEN1 O00255 1/20 0.48
NTSR1 P30989 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20198260 1.00 ALDH1A1 (0.76) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL18652852 0.88 LMNA (0.59) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL9389844 0.87 TPMT (0.65) ALDH1A1LMNASRD5A2SMN1; SMN2TPMT
SCHEMBL1244094 0.87 TPMT (0.65) ALDH1A1LMNASRD5A2SMN1; SMN2TPMT
SCHEMBL3841301 0.87 TPMT (0.65) ALDH1A1LMNASRD5A2SMN1; SMN2TPMT
SCHEMBL822185 0.87 ALDH1A1 (1.00) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL52200 0.87 ALDH1A1 (1.00) ALDH1A1LMNASRD5A2CES2CES1
Hydrochloric Acid SCHEMBL27909743 0.85 ALDH1A1 (0.94) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL11528213 0.85 ALDH1A1 (0.94) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL21230318 0.84 ALDH1A1 (0.54) ALDH1A1LMNASRD5A2CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3350149-B1 [(2-ETHOXY-5-TRANS-1-PROPEN-1-YL)-PHENOXYL]-TERMINATED COMPOUNDS EVONIK DEGUSSA GMBH (DE) 2019-11-20 EP disclosed
EP-2433989-B1 LIGHT-ABSORBING MATERIAL AND PHOTOELECTRIC CONVERSION ELEMENT PANASONIC CORP (JP) 2018-03-14 EP disclosed
EP-3050885-B1 BENZODIAZEPINE BROMODOMAIN INHIBITOR GLAXOSMITHKLINE LLC (US) 2017-10-18 EP disclosed
WO-2017108946-A1 THERMOSETTING RESIN COMPOSITIONS HEXCEL COMPOSITES LIMITED (GB) 2017-06-29 WO disclosed
US-20170145021-A1 NOVEL COMPOUNDS GLAXOSMITHKLINE LLC 2017-05-25 US disclosed
US-20170145021-A1 NOVEL COMPOUNDS GLAXOSMITHKLINE LLC 2017-05-25 US disclosed
WO-2017045931-A1 [(2-ETHOXY-5-TRANS-1-PROPEN-1-YL)-PHENOXYL]-TERMINATED COMPOUNDS EVONIK TECHNOCHEMIE GMBH (DE) 2017-03-23 WO disclosed
EP-3144289-A1 [(2-ETHOXY-5-TRANS-1-PROPEN-1-YL)-PHENOXYL]-TERMINATED COMPOUNDS Evonik Technochemie GmbH (DE) 2017-03-22 EP disclosed
US-9598420-B2 Benzodiazepine bromodomain inhibitor GLAXOSMITHKLINE LLC (US) 2017-03-21 US disclosed
US-9598420-B2 Benzodiazepine bromodomain inhibitor GLAXOSMITHKLINE LLC (US) 2017-03-21 US disclosed
US-20150299210-A1 Benzodiazepine Bromodomain Inhibitor GLAXOSMITHKLINE LLC 2015-10-22 US disclosed
US-20150299210-A1 Benzodiazepine Bromodomain Inhibitor GLAXOSMITHKLINE LLC 2015-10-22 US disclosed
US-9102677-B2 Benzodiazepine bromodomain inhibitor GLAXOSMITHKLINE LLC (US) 2015-08-11 US disclosed
US-9102677-B2 Benzodiazepine bromodomain inhibitor GLAXOSMITHKLINE LLC (US) 2015-08-11 US disclosed
US-20120252781-A1 Benzodiazepine Bromodomain Inhibitor GLAXOSMITHKLINE LLC 2012-10-04 US disclosed
US-20120252781-A1 Benzodiazepine Bromodomain Inhibitor GLAXOSMITHKLINE LLC 2012-10-04 US disclosed
WO-2012001131-A1 METHOD OF MAKING POLY(ARYL ETHER KETONES) FROM 4,4' DIFLUOROBENZOPHENONE COMPRISING OXIDIZING SPECIES AND/OR NITRO COMPOUNDS SOLVAY SPECIALTY POLYMERS USA, L.L.C. (US) 2012-01-05 WO disclosed
WO-2011054845-A1 BENZODIAZEPINE BROMODOMAIN INHIBITOR GLAXOSMITHKLINE LLC (US) 2011-05-12 WO disclosed
US-7927756-B2 Redox fuel cell using methanol FUJITSU LIMITED (JP) 2011-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150299210-A1 Benzodiazepine Bromodomain Inhibitor GABRB1, GABRB3, GABRB2 ALDH1A1 1074/4885LMNA 2329/4885SRD5A2 1449/4885
US-20170145021-A1 NOVEL COMPOUNDS GABRE, GABRA1, GABRA6 ALDH1A1 996/4885LMNA 2687/4885SRD5A2 621/4885
US-20120252781-A1 Benzodiazepine Bromodomain Inhibitor GABRB1, GABRB3, GABRB2 ALDH1A1 1074/4885LMNA 2329/4885SRD5A2 1449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.