SCHEMBL1027753

SCHEMBL1027753

Cc1oc(Cl)nc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HCAR2 Q8TDS4 1/20 0.39
TDP1 Q9NUW8 2/20 0.35
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TARBP2 Q15633 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PDE4B Q07343 1/20 0.32
PIN1 Q13526 1/20 0.32
LMNA P02545 1/20 0.32
RECQL P46063 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GRIA1 P42261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287238 0.77 ALDH1A1 (0.33) ALDH1A1HPGDTSHRHCAR2SMN1; SMN2
Hydrochloric Acid SCHEMBL19119222 0.76 PDE4B (0.33) ALDH1A1HPGDTSHRHCAR2SMN1; SMN2
SCHEMBL13341691 0.74 TARBP2 (0.34) ALDH1A1HPGDTSHRHCAR2SMN1; SMN2
SCHEMBL28775950 0.74 FBP1 (0.51) ALDH1A1TDP1PDE4BPIN1LMNA
SCHEMBL459975 0.74 TDP1 (0.36) ALDH1A1HPGDTSHRHCAR2TDP1
SCHEMBL348144 0.74 HCRTR1 (0.35) ALDH1A1HPGDTSHRHCAR2TARBP2
SCHEMBL29415465 0.73 ALDH1A1 (0.46) ALDH1A1HPGDTSHRHCAR2TDP1
SCHEMBL352388 0.73 ALDH1A1 (0.46) ALDH1A1HPGDTSHRHCAR2TDP1
SCHEMBL9832492 0.71 TARBP2 (0.68) ALDH1A1TDP1SMN1; SMN2TARBP2NPC1
SCHEMBL11173035 0.71 ALDH1A1 (0.45) ALDH1A1HPGDTSHRMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4551571-A1 OXAZOLE TRPML1 AGONISTS AND USES THEREOF Libra Therapeutics, Inc. (US) 2025-05-14 EP disclosed
CN-119790050-A Oxazole TRPML1 agonists and uses thereof 利布拉医疗公司 2025-04-08 CN disclosed
US-12098145-B2 Oxazole TRPML1 agonists and uses thereof LIBRA THERAPEUTICS, INC. (US) 2024-09-24 US disclosed
US-20240158381-A1 OXAZOLE TRPML1 AGONISTS AND USES THEREOF LIBRA THERAPEUTICS, INC. 2024-05-16 US disclosed
WO-2024011155-A1 OXAZOLE TRPML1 AGONISTS AND USES THEREOF LIBRA THERAPEUTICS, INC. (US) 2024-01-11 WO disclosed
WO-2024011155-A1 OXAZOLE TRPML1 AGONISTS AND USES THEREOF LIBRA THERAPEUTICS, INC. (US) 2024-01-11 WO disclosed
US-8513235-B2 Homocysteine synthase inhibitor MITSUBISHI TANABE PHARMA CORPORATION (JP) 2013-08-20 US disclosed
EP-2486925-A1 THERAPEUTIC AGENT FOR CEREBRAL INFARCTION Mitsubishi Tanabe Pharma Corporation (JP) 2012-08-15 EP disclosed
US-20120196824-A1 THERAPEUTIC AGENT FOR CEREBRAL INFARCTION MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-08-02 US disclosed
US-20110034440-A1 HOMOCYSTEINE SYNTHASE INHIBITOR MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-02-10 US disclosed
EP-2275404-A1 HOMOCYSTEINE SYNTHASE INHIBITOR Mitsubishi Tanabe Pharma Corporation (JP) 2011-01-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120196824-A1 THERAPEUTIC AGENT FOR CEREBRAL INFARCTION FABP7, TIMP3, MMP11 ALDH1A1 180/4885HPGD 356/4885TSHR 4241/4885
US-20110034440-A1 HOMOCYSTEINE SYNTHASE INHIBITOR BHMT, CBS, BHMT2 ALDH1A1 600/4885HPGD 222/4885TSHR 2667/4885
US-12098145-B2 Oxazole TRPML1 agonists and uses thereof TRPM7, TRPM2, TRPM5 ALDH1A1 1854/4885HPGD 1075/4885TSHR 1535/4885
US-20240158381-A1 OXAZOLE TRPML1 AGONISTS AND USES THEREOF TRPM7, TRPM2, TRPM5 ALDH1A1 2066/4885HPGD 962/4885TSHR 2320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.