SCHEMBL10539378

SCHEMBL10539378

Nc1ccc(S(=O)(=O)[O-])c2cc(S(=O)(=O)O)cc(O)c12.[Na+]

nearest known ligand 0.57

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.57
NT5E P21589 2/20 0.49
AURKA O14965 1/20 0.49
AURKB Q96GD4 1/20 0.49
HSD17B10 Q99714 3/20 0.49
ALDH1A1 P00352 2/20 0.49
CASP6 P55212 3/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
APEX1 P27695 2/20 0.45
DUSP5 Q16690 1/20 0.43
NSD2 O96028 2/20 0.42
DUSP3 P51452 1/20 0.42
PTPN5 P54829 1/20 0.42
PTPN11 Q06124 1/20 0.42
PTPN1 P18031 2/20 0.41
GAA P10253 2/20 0.40
PLCG1 P19174 1/20 0.40
DNMT1 P26358 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lithium Ion SCHEMBL445794 0.88 NR4A1 (0.60) NR4A1NT5EAURKAAURKBHSD17B10
SCHEMBL156092 0.88 AURKA (0.62) NR4A1NT5EAURKAAURKBHSD17B10
SCHEMBL29706553 0.88 AURKA (0.62) NR4A1NT5EAURKAAURKBHSD17B10
SCHEMBL10539390 0.88 AURKA (0.62) NR4A1NT5EAURKAAURKBHSD17B10
SCHEMBL10539372 0.87 AURKA (0.60) NR4A1NT5EAURKAAURKBHSD17B10
SCHEMBL445795 0.87 AURKA (0.60) NR4A1NT5EAURKAAURKBHSD17B10
Monoethanolamine SCHEMBL10589744 0.81 AURKA (0.54) NR4A1NT5EAURKAAURKBHSD17B10
Aniline SCHEMBL10587235 0.81 AURKA (0.57) NR4A1NT5EAURKAAURKBHSD17B10
SCHEMBL10782044 0.81 NT5E (0.70) NT5EAURKAAURKBHSD17B10ALDH1A1
SCHEMBL15268136 0.80 SENP2 (0.50) NR4A1NT5EAURKAAURKBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4855411-A Water-soluble, monoazo dyes containing a ureido group and two sulfonyl fiber-reactive groups Crall, Hugh C. (US) 1989-08-08 US disclosed