SCHEMBL10694512

SCHEMBL10694512

COc1ccc(C2Cc3ccccc3N(C)C2=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CACNA1S Q13698 5/20 0.51
KMT2A Q03164 3/20 0.48
TSHR P16473 1/20 0.48
PYGL P06737 1/20 0.46
PYGM P11217 1/20 0.46
MEN1 O00255 1/20 0.43
CYP19A1 P11511 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691585 0.85 LMNA (0.49) KMT2ATSHRPYGLPYGMMEN1
SCHEMBL10695532 0.85 TSHR (0.65) KMT2ATSHRPYGLPYGMCYP19A1
SCHEMBL30489285 0.85 TSHR (0.65) KMT2ATSHRPYGLPYGMCYP19A1
SCHEMBL6281661 0.79 CACNA1S (0.53) CACNA1SCYP19A1
SCHEMBL10691415 0.78 DRD2 (0.44) KMT2AMEN1CYP19A1
SCHEMBL6275952 0.77 F10 (0.67) CACNA1S
SCHEMBL9148955 0.74 CYP19A1 (0.59) TSHRCYP19A1
SCHEMBL23959055 0.72 RAB9A (0.51) CACNA1S
SCHEMBL10688450 0.71 ADRA1A (0.46) KMT2ATSHRPYGLPYGM
SCHEMBL9560256 0.71 MAPT (0.56) KMT2APYGLPYGMMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed