SCHEMBL10947765

SCHEMBL10947765

COC(=O)c1cc2c(cc1OCc1ccccc1)CCC/C2=N\O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 3/20 0.46
HPGD P15428 2/20 0.46
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
MAPK1 P28482 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMPD1 P17405 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
RXRA P19793 1/20 0.40
SGMS2 Q8NHU3 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10879814 1.00 ALDH1A1 (0.46) ALDH1A1KDM4EMAPTHPGDMAOA
SCHEMBL10880568 0.86 MAOA (0.58) ALDH1A1KDM4EMAPTHPGDMAOA
SCHEMBL10881146 0.85 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTHPGDMAOA
SCHEMBL10879784 0.83 MAPT (0.55) ALDH1A1KDM4EMAPTHPGDLMNA
SCHEMBL10880892 0.77 RXRA (0.41) ALDH1A1KDM4EMAPTHPGDLMNA
SCHEMBL10880896 0.77 RXRA (0.41) ALDH1A1KDM4EMAPTHPGDLMNA
SCHEMBL8676133 0.77 RXRA (0.42) ALDH1A1KDM4EMAOAMAOBPOLB
SCHEMBL10883172 0.76 FAAH (0.41) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL10881168 0.76 ACHE (0.42) ALDH1A1KDM4EMAPTHPGDMAOA
SCHEMBL9489485 0.76 MAOA (0.66) HPGDMAOAMAOBPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4500545-A HYPOTENSIVE, ANTISECRETORY AGENTS, AND DOPAMINE ANTAGONIST ELI LILLY AND COMPANY (US) 1985-02-19 US disclosed
US-4448990-A Hydroxyaminotetralincarboxamides ELI LILLY AND COMPANY (US) 1984-05-15 US disclosed