SCHEMBL1108476

SCHEMBL1108476

c1ccc(Cc2cocn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 1/20 0.44
ALDH1A1 P00352 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
TAAR1 Q96RJ0 1/20 0.37
LMNA P02545 1/20 0.37
HTR2B P41595 1/20 0.37
AOC3 Q16853 1/20 0.35
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
MAOB P27338 1/20 0.35
SCN9A Q15858 1/20 0.34
KAT7 O95251 1/20 0.34
KAT6A Q92794 1/20 0.34
SORT1 Q99523 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29084377 0.82 KCNH2 (0.50) ALDH1A1SMN1; SMN2TDP1TAAR1HPGD
SCHEMBL29348977 0.80 ESR1 (0.48) TAAR1
SCHEMBL12848465 0.78 TAAR1 (0.41) ALDH1A1SMN1; SMN2TDP1TAAR1HTR2B
SCHEMBL16598215 0.76 L3MBTL1 (0.44) ALDH1A1SMN1; SMN2L3MBTL1TDP1TAAR1
SCHEMBL12794242 0.76 KAT7 (0.39) ALDH1A1SMN1; SMN2TDP1HPGDTSHR
SCHEMBL17239520 0.71 PDE10A (0.46) ALDH1A1L3MBTL1HPGDTSHRSCN9A
SCHEMBL27072915 0.70 CALM1 (0.55) CALM1ALDH1A1RAB9ASMN1; SMN2L3MBTL1
Hydrochloric Acid SCHEMBL4829192 0.69 HIF1A (0.39) ALDH1A1TSHR
SCHEMBL64435 0.67 L3MBTL1 (0.68) CALM1ALDH1A1RAB9ASMN1; SMN2L3MBTL1
SCHEMBL415622 0.67 CALM1 (0.50) CALM1ALDH1A1RAB9ASMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4142732-B1 METHODS OF USE FOR PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS INC (US) 2026-04-22 EP disclosed
US-12016312-B2 Animal models, screening methods, and treatment methods for intraocular diseases or disorders Smilebiotek Zhuhai Limited (CN) 2024-06-25 US disclosed
CN-110267960-A Substituted pyrazolo [1,5-a] pyrazine compound as RET kinase inhibitor 阿雷生物药品公司 2019-09-20 CN disclosed
CN-105658642-B Fibroblast growth factor receptor inhibitors 蓝图药品公司 2019-05-03 CN disclosed
CN-103826661-B Novel binding agent-drug conjugates (ADCs) and uses thereof 西雅图基因公司 2019-03-05 CN disclosed
CN-108193309-A Ultra-fine denier polyester filament yarn and preparation method thereof 海盐县硕创服装研究所 2018-06-22 CN disclosed
CN-107849010-A 3, 3-difluoropiperidine carbamate heterocycles as NR2B NMDA receptor antagonists 卢郡控股(开曼)有限公司 2018-03-27 CN disclosed
US-8153673-B2 Metalloproteinase inhibitors ASTRAZENECA AB (SE) 2012-04-10 US disclosed
US-20110003853-A1 Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2011-01-06 US disclosed
US-20100273849-A1 Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2010-10-28 US disclosed
US-20080262045-A1 Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2008-10-23 US disclosed
US-7427631-B2 especially as inhibitors of MMP12 ASTRAZENECA AB (SE) 2008-09-23 US disclosed
US-20080171882-A1 Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2008-07-17 US disclosed
US-7368465-B2 Respiratory system disorders; antiarthritic agents; anticancer agents; bone disorders ASTRAZENECA AB (SE) 2008-05-06 US disclosed
US-20040138276-A1 Metalloproteinase inhibitors ASTRAZENECA AB (SE) 2004-07-15 US disclosed
US-5968725-A MATERIAL COMPRISING ON SUPPORT SILVER HALIDE PHOTOSENSITIVE LAYER CONTAINING ORGANIC SILVER SALT, REDUCING AGENT, ULTRAHIGH CONTRAST PROMOTING AGENT, SELECTED HETEROCYCLIC MERCAPTO COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 1999-10-19 US disclosed
EP-0385999-A1 APPLICATION OF 4- 1-OXOALKYL]-2,5-OXAZOLIDINEDIONES IN SELECTIVE STEREOSPECIFIC FORMATION OF BIOLOGICALLY ACTIVE BETA-LACTAMS. UNIV CINCINNATI (US) 1990-09-12 EP disclosed
WO-1988010256-A1 APPLICATION OF 4-[1-OXOALKYL]-2,5-OXAZOLIDINEDIONES IN SELECTIVE STEREOSPECIFIC FORMATION OF BIOLOGICALLY ACTIVE BETA-LACTAMS UNIVERSITY OF CINCINNATI (US) 1988-12-29 WO disclosed
US-4769316-A Method for restraining the formation of re-reversal negative image in direct positive silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1988-09-06 US disclosed
US-4607006-A Silver halide photographic light-sensitive material containing non-spectral sensitizing electron donative silver halide adsorptive compound FUJI PHOTO FILM CO., LTD. (JP) 1986-08-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110003853-A1 Metalloproteinase Inhibitors MMP9, MMP12, MMP14 CALM1 2925/4885ALDH1A1 612/4885RAB9A 2412/4885
US-20100273849-A1 Metalloproteinase Inhibitors MMP9, MMP12, MMP11 CALM1 2829/4885ALDH1A1 1381/4885RAB9A 1625/4885
US-20080171882-A1 Metalloproteinase Inhibitors MMP9, MMP12, MMP14 CALM1 2925/4885ALDH1A1 612/4885RAB9A 2412/4885
US-20080262045-A1 Metalloproteinase Inhibitors MMP9, MMP12, MMP11 CALM1 2829/4885ALDH1A1 1381/4885RAB9A 1625/4885
US-12016312-B2 Animal models, screening methods, and treatment methods for intraocular diseases or disorders MB, MYOC, PDE6A CALM1 3826/4885ALDH1A1 1091/4885RAB9A 1921/4885
US-20040138276-A1 Metalloproteinase inhibitors MMP9, MMP11, MMP7 CALM1 2737/4885ALDH1A1 1172/4885RAB9A 1251/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.