SCHEMBL1189696

SCHEMBL1189696

CN1C(=O)CN(Cc2ccccc2)C(=O)C12CC2

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.48
KMT2A Q03164 6/20 0.48
ELANE P08246 2/20 0.42
EPHX2 P34913 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
DDB1 Q16531 1/20 0.42
CRBN Q96SW2 1/20 0.42
DRD3 P35462 1/20 0.40
KCNH2 Q12809 1/20 0.40
ENPP2 Q13822 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
ACHE P22303 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21228482 0.78 KMT2A (0.50) MEN1KMT2AELANEEPHX2L3MBTL1
SCHEMBL1488276 0.74 L3MBTL1 (0.56) MEN1KMT2AELANEEPHX2L3MBTL1
SCHEMBL21228493 0.73 KMT2A (0.51) MEN1KMT2AELANEEPHX2L3MBTL1
SCHEMBL16085590 0.72 KMT2A (0.49) MEN1KMT2AEPHX2L3MBTL1DDB1
SCHEMBL7212064 0.72 ENPP2 (0.53) MEN1KMT2AELANEEPHX2L3MBTL1
SCHEMBL24992399 0.71 KMT2A (0.61) MEN1KMT2AELANEEPHX2L3MBTL1
SCHEMBL1189753 0.71 KMT2A (0.61) MEN1KMT2AELANEEPHX2L3MBTL1
SCHEMBL3207582 0.71 ELANE (0.56) MEN1KMT2AELANEEPHX2L3MBTL1
SCHEMBL21228094 0.71 RIPK1 (0.49) MEN1KMT2AELANEDDB1CRBN
SCHEMBL21228083 0.71 GAA (0.48) MEN1KMT2AELANEDDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217226-B1 PEPTIDE DEFORMYLASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2015-07-22 EP disclosed
US-20130045962-A1 PEPTIDE DEFORMYLASE INHIBITORS GLAXOSMITHKLINE LLC 2013-02-21 US disclosed
US-7893056-B2 Peptide deformylase inhibitors GLAXOSMITHKLINE LLC (US) 2011-02-22 US disclosed
EP-2217226-A1 PEPTIDE DEFORMYLASE INHIBITORS GlaxoSmithKline LLC (US) 2010-08-18 EP disclosed
US-20090306066-A1 PEPTIDE DEFORMYLASE INHIBITORS GLAXOSMITHKLINE LLC 2009-12-10 US disclosed
WO-2009061879-A1 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-05-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130045962-A1 PEPTIDE DEFORMYLASE INHIBITORS PDF, DPEP1, DHPS MEN1 2465/4885KMT2A 1907/4885ELANE 451/4885
US-20090306066-A1 PEPTIDE DEFORMYLASE INHIBITORS PDF, DHPS, PADI3 MEN1 3499/4885KMT2A 2169/4885ELANE 498/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.