SCHEMBL12366170

SCHEMBL12366170

[C-]#[N+]CC(=O)NCc1cc(F)ccc1F

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.46
ALDH1A1 P00352 3/20 0.46
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.45
MAPK8 P45983 1/20 0.41
ERCC1 P07992 1/20 0.40
ERCC4 Q92889 1/20 0.40
RAB9A P51151 1/20 0.40
P2RX7 Q99572 2/20 0.39
MET P08581 1/20 0.38
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
CHRM4 P08173 1/20 0.38
TRPV1 Q8NER1 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366137 0.88 P2RX7 (0.50) MAPK8ERCC1ERCC4RAB9AP2RX7
SCHEMBL12366210 0.83 ERCC1 (0.40) ALDH1A1MAPTERCC1ERCC4RAB9A
SCHEMBL12366161 0.82 RIPK1 (0.38) P2RX7ROCK2ROCK1CHRM4
SCHEMBL12366133 0.81 HPGD (0.54) ALDH1A1LMNAMAPTRAB9ASMN1; SMN2
SCHEMBL12366166 0.80 P2RX7 (0.49) P2RX7
SCHEMBL4033108 0.80 CNR1 (0.52) CNR1ALDH1A1LMNAMAPTMAPK8
SCHEMBL12366135 0.78 LMNA (0.62) ALDH1A1LMNARAB9ASMN1; SMN2
SCHEMBL3562274 0.77 ALDH1A1 (0.48) CNR1ALDH1A1LMNAMAPTMAPK8
SCHEMBL14393385 0.77 LMNA (0.52) CNR1ALDH1A1LMNAMAPT
SCHEMBL12366168 0.77 P2RX7 (0.44) ALDH1A1LMNAP2RX7TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed