SCHEMBL12499730

SCHEMBL12499730

COC(=O)c1c(Cc2ccc(Cl)c(Cl)c2)nn(C)c1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
MAPT P10636 3/20 0.42
FPR2 P25090 2/20 0.41
PROKR1 Q8TCW9 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
NOTUM Q6P988 1/20 0.40
ALDH1A1 P00352 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 2/20 0.38
RAB9A P51151 1/20 0.38
PLA2G2A P14555 1/20 0.38
P2RX7 Q99572 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12499672 0.86 RNASEH1 (0.43) MAPTFPR2PROKR1KMT2AGAA
SCHEMBL12499862 0.86 PLA2G2A (0.45) MAPTSMN1; SMN2ALDH1A1L3MBTL1KMT2A
SCHEMBL12498726 0.84 HSP90AA1 (0.47) MAPTSMN1; SMN2ALDH1A1KMT2AGAA
SCHEMBL12498677 0.81 PLA2G2A (0.45) MAPTSMN1; SMN2ALDH1A1KMT2AGAA
SCHEMBL3718927 0.81 ALDH1A1 (0.47) TSHRMAPTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL12499839 0.78 LMNA (0.43) MAPTALDH1A1KMT2AGAAKDM4E
SCHEMBL12499851 0.77 ALDH1A1 (0.43) MAPTSMN1; SMN2ALDH1A1L3MBTL1KMT2A
SCHEMBL12498769 0.77 GPR52 (0.44) MAPTSMN1; SMN2KMT2AKDM4E
SCHEMBL12499589 0.75 ALOX5 (0.43) TSHRMAPTSMN1; SMN2NOTUMALDH1A1
SCHEMBL12499826 0.72 CCR2 (0.39) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012103071-A2 COMPOUNDS AND COMPOSITIONS EISAI R&D MANAGEMENT CO., LTD. (JP) 2012-08-02 WO disclosed