SCHEMBL12866893

SCHEMBL12866893

CC(C)Oc1cccc(CC(C)(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.46
P2RX3 P56373 1/20 0.44
TAAR1 Q96RJ0 2/20 0.42
CETP P11597 2/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
FFAR4 Q5NUL3 2/20 0.40
KDM4E B2RXH2 2/20 0.39
NSD2 O96028 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HSD17B10 Q99714 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
SLC13A5 Q86YT5 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18014708 0.90 RXRA (0.50) DHFRP2RX3RXRARXRBFFAR4
SCHEMBL15356485 0.85 GPBAR1 (0.42) TAAR1HSD17B10GAAPPARGPPARA
SCHEMBL12866847 0.85 GPBAR1 (0.42) TAAR1HSD17B10GAAPPARGPPARA
SCHEMBL1690345 0.84 MEP1B (0.47) TAAR1CETPKDM4EHCRTR1HCRTR2
SCHEMBL12881236 0.80 ALOX5 (0.49) DHFRP2RX3TAAR1FFAR4PPARG
SCHEMBL25053658 0.80 MTNR1A (0.42)
SCHEMBL25053662 0.80 MTNR1A (0.42)
SCHEMBL1908523 0.79 MAPK1 (0.49) DHFRP2RX3TAAR1RXRARXRB
SCHEMBL73635 0.79 TAAR1 (0.56) TAAR1ALDH1A1
SCHEMBL278395 0.79 FAAH (0.42) TAAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9561212-B2 Hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2017-02-07 US disclosed
US-20130150376-A1 Novel Sultam Compounds PFIZER INC. (US) 2013-06-13 US disclosed
US-20110046160-A1 Novel Class of Spiro Piperidines for the Treatment of Neurodegenerative Diseases PFIZER, INC. 2011-02-24 US disclosed
US-20100216796-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS KATTAR SOLOMON 2010-08-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100216796-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS BRDT, AADAC, ACIN1 DHFR 717/4885P2RX3 2867/4885TAAR1 1858/4885
US-20130150376-A1 Novel Sultam Compounds SULT2A1, SULT1A1, SULT1E1 DHFR 316/4885P2RX3 2674/4885TAAR1 1314/4885
US-20110046160-A1 Novel Class of Spiro Piperidines for the Treatment of Neurodegenerative Diseases SNCA, PARK7, HTT DHFR 89/4885P2RX3 651/4885TAAR1 522/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.