SCHEMBL13415

SCHEMBL13415

Brc1ccc2n[nH]cc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.44
CSNK2A1 P68400 2/20 0.39
NOS1 P29475 2/20 0.39
METAP2 P50579 2/20 0.39
PABPC1 P11940 1/20 0.38
CYP2A6 P11509 2/20 0.38
ALDH1A1 P00352 2/20 0.38
AHR P35869 1/20 0.38
NR4A2 P43354 1/20 0.38
CASP3 P42574 1/20 0.38
TYMS P04818 1/20 0.37
ILK Q13418 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
HTT P42858 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
DYRK1A Q13627 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25207842 0.83 BACE1 (0.45) BACE1CSNK2A1NOS1METAP2PABPC1
SCHEMBL12653740 0.76 CYP1A2 (0.48) BACE1CYP2A6ALDH1A1KDM4EMEN1
SCHEMBL19359062 0.74 ALDH1A1 (0.48) ALDH1A1KDM4EMEN1KMT2AHTT
SCHEMBL16523221 0.74 F7 (0.48) BACE1NOS1CYP2A6ALDH1A1AHR
SCHEMBL16523329 0.74 BACE1 (0.44) BACE1CYP2A6ALDH1A1AHRCASP3
SCHEMBL4773397 0.74 NOS1 (0.39) NOS1TYMSMAPT
SCHEMBL18003378 0.71 KDM4E (0.50) CYP2A6ALDH1A1KDM4EMEN1KMT2A
SCHEMBL23786 0.71 ENPP2 (0.46)
SCHEMBL17127346 0.69 SCN10A (0.44) CSNK2A1METAP2ALDH1A1KMT2ADYRK1A
SCHEMBL25422558 0.69 ALDH1A1 (0.37) ALDH1A1MEN1MAPTKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4611899-A1 ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASE Petra Pharma Corporation (US) 2025-09-10 EP disclosed
EP-4598923-A1 SUPRAMOLECULAR POLYMER THERAPEUTICS AND DIAGNOSTICS The Regents of the University of California (US) 2025-08-13 EP disclosed
US-20250082633-A1 COMPOUNDS AND METHODS FOR MODULATING SPLICING REMIX THERAPEUTICS INC (US) 2025-03-13 US disclosed
WO-2025049746-A1 COMPOSITIONS COMPRISING WERNER SYNDROME HELICASE INHIBITORS AND METHODS OF USING THE SAME EIKON THERAPEUTICS, INC. (US) 2025-03-06 WO disclosed
WO-2025021182-A1 CYP11A1 INHIBITORS ACERAND THERAPEUTICS (HONG KONG) LIMITED (CN) 2025-01-30 WO disclosed
CN-118804912-A Compounds and methods for modulating splicing 雷密克斯医疗公司 2024-10-18 CN disclosed
EP-4436961-A1 COMPOUNDS AND METHODS FOR MODULATING SPLICING Remix Therapeutics Inc. (US) 2024-10-02 EP disclosed
WO-2024182778-A1 COMPOUNDS AND METHODS FOR MODULATING SPLICING REMIX THERAPEUTICS INC. (US) 2024-09-06 WO disclosed
US-20240287063-A1 METHIONINE ADENOSYLTRANSFERASE 2A INHIBITOR NANJING CHIA TAI TIANQING PHARMACEUTICAL CO., LTD. (CN) 2024-08-29 US disclosed
US-20240199604-A1 SUPRAMOLECULAR POLYMER THERAPEUTICS AND DIAGNOSTICS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-06-20 US disclosed
US-20090264406-A1 3-METHYL-IMIDAZO[1,2-B]PYRIDAZINE DERIVATIVES NOVARTIS AG 2009-10-22 US disclosed
WO-2009106577-A1 IMIDAZO [1,2-B] PYRIDAZINE DERIVATIVES FOR THE TREATMENT OF C-MET TYROSINE KINASE MEDIATED DISEASE NOVARTIS AG (CH) 2009-09-03 WO disclosed
CN-1243723-C N-phenylpropylcyclopentyl substituted glutaramide derivatives as NEP inhibitors of FSAD PFIZER LTD (US) 2006-03-01 CN disclosed
US-6849649-B2 N-phenpropylcyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase PFIZER INC. (US) 2005-02-01 US disclosed
US-20040106611-A1 N-phenpropylcyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase PFIZER INC 2004-06-03 US disclosed
CN-1492852-A N-phenylpropylcyclopentyl substituted glutaramide derivatives as NEP inhibitors of FSAD ������ҩ�����޹�˾ 2004-04-28 CN disclosed
EP-1373192-A1 N-PHENPROPYLCYCLOPENTYL-SUBSTITUTED GLUTARAMIDE DERIVATIVES AS NEP INHIBITORS FOR FSAD Pfizer Limited (GB) 2004-01-02 EP disclosed
US-6660756-B2 N-phenpropylcyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase PFIZER INC. 2003-12-09 US disclosed
US-20030105132-A1 N-phenpropylcuclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase PFIZER INC. 2003-06-05 US disclosed
WO-2002079143-A1 N-PHENPROPYLCYCLOPENTYL-SUBSTITUTED GLUTARAMIDE DERIVATIVES AS NEP INHIBITORS FOR FSAD PFIZER LIMITED (GB) 2002-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240199604-A1 SUPRAMOLECULAR POLYMER THERAPEUTICS AND DIAGNOSTICS MAPT, HTT, PSEN1 BACE1 27/4885CSNK2A1 2137/4885NOS1 4315/4885
US-20250082633-A1 COMPOUNDS AND METHODS FOR MODULATING SPLICING RBM17, SNRPA, SNRPA1 BACE1 668/4885CSNK2A1 1877/4885NOS1 1941/4885
US-20240287063-A1 METHIONINE ADENOSYLTRANSFERASE 2A INHIBITOR MAT2A, MAT2B, MAT1A BACE1 1850/4885CSNK2A1 3367/4885NOS1 1258/4885
US-20090264406-A1 3-METHYL-IMIDAZO[1,2-B]PYRIDAZINE DERIVATIVES MET, ERBB2, ALK BACE1 4082/4885CSNK2A1 78/4885NOS1 2248/4885
US-20030105132-A1 N-phenpropylcuclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase PREP, ENGASE, ENPEP BACE1 829/4885CSNK2A1 2786/4885NOS1 1287/4885
US-20040106611-A1 N-phenpropylcyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase PREP, ENGASE, ENPEP BACE1 1072/4885CSNK2A1 2915/4885NOS1 1205/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.