SCHEMBL1344286

SCHEMBL1344286

CCC(c1ccccc1)C(C#N)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.68
ESR2 Q92731 4/20 0.68
TRPA1 O75762 2/20 0.47
HKDC1 Q2TB90 1/20 0.46
LMNA P02545 3/20 0.42
TSHR P16473 1/20 0.42
MAP2K1 Q02750 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
MIF P14174 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A3 Q01959 2/20 0.38
MAPT P10636 2/20 0.38
ALOX15 P16050 2/20 0.38
CYP1A2 P05177 1/20 0.38
PGR P06401 1/20 0.38
CHRM2 P08172 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
AR P10275 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17947359 0.85 ESR1 (0.50) ESR1ESR2TRPA1HKDC1LMNA
SCHEMBL24849087 0.82 TRPA1 (0.48) ESR1ESR2TRPA1HKDC1LMNA
SCHEMBL4413894 0.80 ESR1 (0.44) ESR1ESR2TRPA1LMNATSHR
SCHEMBL28981577 0.78 ESR1 (0.47) ESR1ESR2TRPA1LMNATSHR
SCHEMBL819626 0.78 ESR1 (0.56) ESR1ESR2TRPA1LMNATSHR
SCHEMBL6309534 0.78 ESR1 (0.56) ESR1ESR2TRPA1LMNATSHR
SCHEMBL4071581 0.78 HKDC1 (0.65) ESR1TRPA1HKDC1LMNATAAR1
SCHEMBL17702682 0.77 ESR1 (0.46) ESR1ESR2TRPA1HKDC1LMNA
SCHEMBL17702681 0.77 ESR1 (0.46) ESR1ESR2TRPA1HKDC1LMNA
SCHEMBL28979280 0.77 TRPA1 (0.44) ESR1ESR2TRPA1HKDC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10172350-B2 Substituted 5-hydroxy-2-phenyl-3-heteroaryl pentanenitrile derivatives, method for the production thereof and use thereof as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-01-08 US disclosed
US-10021877-B2 Substituted 5-hydroxy-2,3-diphenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-07-17 US disclosed
US-9957248-B2 Substituted 5-hydroxy-2-heteroaryl-3-phenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSHAFT (DE) 2018-05-01 US disclosed
EP-3003036-B1 SUBSTITUTED 5-HYDROXY-2,3-DIPHENYLPENTANONITRILE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2018-04-11 EP disclosed
US-20170290330-A1 SUBSTITUTED 5-HYDROXY-2-PHENYL-3-HETEROARYL PENTANENITRILE DERIVATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND/OR PLANT GROWH REGULATORS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2017-10-12 US disclosed
CN-107001313-A Substituted 5-hydroxy-2-phenyl-3-heteroarylvaleronitrile derivatives, method for the production thereof and use thereof as herbicides and/or plant growth regulators 拜耳作物科学股份公司 2017-08-01 CN disclosed
US-20170166549-A1 Substituted 5-hydroxy-2-heteroaryl-3-phenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSHAFT (DE) 2017-06-15 US disclosed
CN-106795113-A The phenyl pentane nitrile derivative of 5 hydroxyl, 2 heteroaryl 3 of substitution, its preparation method and its as herbicide and/or the purposes of plant growth regulator 拜耳作物科学股份公司 2017-05-31 CN disclosed
CN-103748075-B 2,3-diphenyl valeronitrile derivant, its preparation method and as herbicide and the purposes of plant growth regulator 拜耳知识产权有限责任公司 2016-09-07 CN disclosed
CN-103748075-B 2,3-diphenyl valeronitrile derivant, its preparation method and as herbicide and the purposes of plant growth regulator 拜耳知识产权有限责任公司 2016-09-07 CN disclosed
WO-2009085072-A1 COMPOSITION COMPRISING CHELATING AGENTS CONTAINING AMIDOXIME COMPOUNDS EKC TECHNOLOGY, INC (US) 2009-07-09 WO disclosed
US-20090137191-A1 COPPER CMP POLISHING PAD CLEANING COMPOSITION COMPRISING OF AMIDOXIME COMPOUNDS EKC TECHNOLOGY, INC. 2009-05-28 US disclosed
US-20090133716-A1 METHODS OF POST CHEMICAL MECHANICAL POLISHING AND WAFER CLEANING USING AMIDOXIME COMPOSITIONS EKC TECHNOLOGY, INC. 2009-05-28 US disclosed
US-20090130849-A1 CHEMICAL MECHANICAL POLISHING AND WAFER CLEANING COMPOSITION COMPRISING AMIDOXIME COMPOUNDS AND ASSOCIATED METHOD FOR USE EKC TECHNOLOGY, INC. 2009-05-21 US disclosed
WO-2009058274-A1 CHEMICAL MECHANICAL POLISHING AND WAFER CLEANING COMPOSITION COMPRISING AMIDOXIME COMPOUNDS AND ASSOCIATED METHOD FOR USE EKC TECHNOLOGY, INC. (US) 2009-05-07 WO disclosed
WO-2009058272-A1 COPPER CMP POLISHING PAD CLEANING COMPOSITION COMPRISING OF AMIDOXIME COMPOUNDS EKC TECHNOLOGY, INC. (US) 2009-05-07 WO disclosed
WO-2009058288-A1 AMIDOXIME COMPOUNDS AS CHELATING AGENTS IN SEMICONDUCTOR PROCESSES EKC TECHNOLOGY, INC. (US) 2009-05-07 WO disclosed
WO-2009058275-A1 METHODS OF POST CHEMICAL MECHANICAL POLISHING AND WAFER CLEANING USING AMIDOXIME COMPOSITIONS EKC TECHNOLOGY, INC. (US) 2009-05-07 WO disclosed
WO-2009058278-A1 METHODS OF CLEANING SEMICONDUCTOR DEVICES AT THE BACK END OF LINE USING AMIDOXIME COMPOSITIONS EKC TECHNOLOGY, INC (US) 2009-05-07 WO disclosed
US-20090107520-A1 AMIDOXIME COMPOUNDS AS CHELATING AGENTS IN SEMICONDUCTOR PROCESSES EKC TECHNOLOGY, INC. 2009-04-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10172350-B2 Substituted 5-hydroxy-2-phenyl-3-heteroaryl pentanenitrile derivatives, method for the production thereof and use thereof as herbicides and/or plant growth regulators HPD, HAAO, GRHPR ESR1 4792/4885ESR2 4043/4885TRPA1 4593/4885
US-10021877-B2 Substituted 5-hydroxy-2,3-diphenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators HPD, DDT, HDHD5 ESR1 4570/4885ESR2 3421/4885TRPA1 4238/4885
US-20090137191-A1 COPPER CMP POLISHING PAD CLEANING COMPOSITION COMPRISING OF AMIDOXIME COMPOUNDS PADI2, PADI4, PADI3 ESR1 4127/4885ESR2 4226/4885TRPA1 3045/4885
US-20170290330-A1 SUBSTITUTED 5-HYDROXY-2-PHENYL-3-HETEROARYL PENTANENITRILE DERIVATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND/OR PLANT GROWH REGULATORS HPD, GRHPR, PAH ESR1 4793/4885ESR2 4020/4885TRPA1 4675/4885
US-20170166549-A1 Substituted 5-hydroxy-2-heteroaryl-3-phenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators HPD, PAH, DDT ESR1 4724/4885ESR2 4086/4885TRPA1 4603/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.