SCHEMBL13628824

SCHEMBL13628824

COOSc1ccc2c(c1)cc(-c1nnco1)n2Cc1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.36
NPC1 O15118 1/20 0.36
PTGS2 P35354 2/20 0.36
NOTUM Q6P988 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
TBXA2R P21731 2/20 0.33
S1PR3 Q99500 1/20 0.32
TRPC5 Q9UL62 1/20 0.32
P2RX7 Q99572 2/20 0.31
ALOX5AP P20292 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
TNIK Q9UKE5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628861 0.85 RAB9A (0.38) RAB9ANPC1NOTUMTSHRMAPK1
SCHEMBL13628851 0.82 PTGS2 (0.36) PTGS2TSHRTBXA2RALDH1A1HTT
SCHEMBL13628832 0.80 TRPC5 (0.38) RAB9ANPC1PTGS2TSHRMAPK1
SCHEMBL13628859 0.80 PTGS2 (0.45) PTGS2TBXA2RPOLB
SCHEMBL13628853 0.79 PTGS2 (0.37) PTGS2TSHRTBXA2RALDH1A1MAPT
SCHEMBL2925335 0.78 PTGS2 (0.56) RAB9ANPC1PTGS2NOTUMTSHR
SCHEMBL13628850 0.77 PTGS2 (0.36) RAB9APTGS2TSHRTBXA2RMAPT
SCHEMBL13628847 0.77 CYP11B2 (0.43) PTGS2MAPT
SCHEMBL13628821 0.77 MAPT (0.37) RAB9APTGS2TSHRMAPK1TBXA2R
SCHEMBL13628857 0.77 CCR2 (0.40) PTGS2TSHRTBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed