SCHEMBL13628859

SCHEMBL13628859

COOSc1ccc2c(c1)cc(-c1ccncc1)n2Cc1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.45
PDE5A O76074 1/20 0.37
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
NFATC1 O95644 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
GNRHR P30968 1/20 0.35
TBXA2R P21731 1/20 0.34
RIPK3 Q9Y572 2/20 0.34
ACLY P53396 1/20 0.34
KCNK13 Q9HB14 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628847 0.88 CYP11B2 (0.43) PTGS2GNRHRACLY
SCHEMBL13628860 0.85 PTGS2 (0.46) PTGS2TP53GNRHRTBXA2R
SCHEMBL13628821 0.82 MAPT (0.37) PTGS2TP53TBXA2R
SCHEMBL13628848 0.81 PTGS2 (0.42) PTGS2GNRHR
SCHEMBL13628853 0.81 PTGS2 (0.37) PTGS2TBXA2R
SCHEMBL13628850 0.80 PTGS2 (0.36) PTGS2TBXA2R
SCHEMBL13628824 0.80 RAB9A (0.36) PTGS2POLBTBXA2R
SCHEMBL13628851 0.80 PTGS2 (0.36) PTGS2TP53TBXA2R
SCHEMBL13628832 0.79 TRPC5 (0.38) PTGS2POLB
SCHEMBL13628857 0.78 CCR2 (0.40) PTGS2TP53TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed