SCHEMBL13628851

SCHEMBL13628851

COOSc1ccc2c(c1)cc(-c1nc(C)no1)n2Cc1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.36
DRD2 P14416 1/20 0.35
SCARB1 Q8WTV0 5/20 0.35
P2RX3 P56373 1/20 0.34
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 2/20 0.33
KMT2A Q03164 2/20 0.33
KCNH2 Q12809 1/20 0.33
MEN1 O00255 1/20 0.33
TP53 P04637 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TBXA2R P21731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628853 0.85 PTGS2 (0.37) PTGS2DRD2ALDH1A1HTTKMT2A
SCHEMBL13628824 0.82 RAB9A (0.36) PTGS2ALDH1A1HTTTSHRTBXA2R
SCHEMBL13628850 0.80 PTGS2 (0.36) PTGS2GRIN1GRIN2BHTTKMT2A
SCHEMBL13628859 0.80 PTGS2 (0.45) PTGS2TP53TBXA2R
SCHEMBL13628821 0.78 MAPT (0.37) PTGS2ALDH1A1KMT2AMEN1TP53
SCHEMBL2928583 0.78 PTGS2 (0.56) PTGS2SCARB1TBXA2R
SCHEMBL13628832 0.78 TRPC5 (0.38) PTGS2ALDH1A1HTTKMT2AMEN1
SCHEMBL13628857 0.77 CCR2 (0.40) PTGS2TP53TSHRNPSR1TBXA2R
SCHEMBL13628847 0.77 CYP11B2 (0.43) PTGS2NPSR1
SCHEMBL13628860 0.76 PTGS2 (0.46) PTGS2TP53TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed