SCHEMBL13628841

SCHEMBL13628841

COOSc1ccc2c(c1)cc(-c1ccc(C(=O)OC)cn1)n2Cc1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 4/20 0.42
LMNA P02545 3/20 0.42
P2RX3 P56373 2/20 0.40
F10 P00742 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
KMT2A Q03164 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
THRB P10828 1/20 0.36
GABRA5 P31644 1/20 0.35
HTT P42858 1/20 0.35
PTGS2 P35354 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628843 0.92 AGTR1 (0.40) TP53POLBPTGS2
SCHEMBL13628844 0.91 TP53 (0.37) TP53POLBMAPTLMNAPTGS2
SCHEMBL2922490 0.83 PTGS2 (0.54) TP53POLBMAPTLMNAP2RX3
SCHEMBL13628857 0.76 CCR2 (0.40) TP53LMNAKDM4EPTGS2
SCHEMBL13628859 0.75 PTGS2 (0.45) TP53POLBPTGS2
SCHEMBL13628853 0.75 PTGS2 (0.37) MAPTLMNAKDM4EALDH1A1KMT2A
SCHEMBL2925431 0.75 PTGS2 (0.48) POLBMAPTLMNAF10KDM4E
SCHEMBL13628821 0.74 MAPT (0.37) TP53MAPTLMNAKDM4EALDH1A1
SCHEMBL13628847 0.74 CYP11B2 (0.43) MAPTPTGS2
SCHEMBL2921231 0.73 PTGS2 (0.52) TP53PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed