SCHEMBL13628852

SCHEMBL13628852

COOSc1ccc2c(c1)cc(C1CCOCC1)n2Cc1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 6/20 0.39
PDE1B Q01064 6/20 0.39
PDE1C Q14123 6/20 0.39
PDE2A O00408 2/20 0.39
HRH1 P35367 4/20 0.37
CYP2D6 P10635 3/20 0.37
CHRM1 P11229 2/20 0.37
PDE10A Q9Y233 1/20 0.36
KCNH2 Q12809 2/20 0.35
PTGS2 P35354 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
PDE9A O76083 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
HSD17B10 Q99714 1/20 0.33
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
CCR2 P41597 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628839 0.85 PDE2A (0.34) PDE1APDE1BPDE1CPDE2AHRH1
SCHEMBL13176309 0.79 PDE1A (0.42) PDE1APDE1BPDE1CPDE2AHRH1
SCHEMBL2920935 0.78 PTGS2 (0.49) PDE1APDE1BPDE1CPDE2AHRH1
SCHEMBL13628840 0.76 PTGS2 (0.35) PTGS2CCR2
SCHEMBL13628832 0.73 TRPC5 (0.38) PTGS2CNR1CNR2HSD17B10
SCHEMBL13628859 0.72 PTGS2 (0.45) PTGS2
SCHEMBL13628853 0.72 PTGS2 (0.37) PTGS2
SCHEMBL13628857 0.71 CCR2 (0.40) PTGS2CCR2
SCHEMBL13628824 0.71 RAB9A (0.36) PTGS2
SCHEMBL13628847 0.69 CYP11B2 (0.43) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed