SCHEMBL14636309

SCHEMBL14636309

COc1ccc(S(=O)(=O)NC#CC[C@@H](C(=O)NOC(C)(C)C)C(C)C)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
MMP13 P45452 12/20 0.41
MMP2 P08253 11/20 0.41
MMP1 P03956 8/20 0.41
MMP9 P14780 8/20 0.41
MMP8 P22894 7/20 0.41
MMP3 P08254 6/20 0.41
MMP7 P09237 2/20 0.41
HSD17B10 Q99714 2/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
MMP14 P50281 2/20 0.38
ADAM17 P78536 1/20 0.38
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14636108 0.87 MMP13 (0.52) MMP13MMP2MMP1MMP9MMP8
SCHEMBL14636268 0.84 MMP2 (0.51) SLC1A3SLC1A2SLC1A1MMP13MMP2
SCHEMBL7305749 0.72 MMP13 (0.71) SLC1A3SLC1A2SLC1A1MMP13MMP2
SCHEMBL7344506 0.71 SLC1A3 (0.56) SLC1A3SLC1A2SLC1A1MMP13MMP2
SCHEMBL7344510 0.71 SLC1A3 (0.56) SLC1A3SLC1A2SLC1A1MMP13MMP2
SCHEMBL7301899 0.68 MMP1 (0.49) MMP13MMP2MMP1MMP9MMP8
SCHEMBL7312224 0.65 ADAM17 (0.48) MMP13MMP2MMP1MMP3HSD17B10
SCHEMBL7892155 0.64 ALDH1A1 (0.66) SLC1A3SLC1A2SLC1A1MMP13MMP2
SCHEMBL7087648 0.64 MMP9 (0.64) SLC1A3SLC1A2SLC1A1MMP13MMP2
SCHEMBL5093836 0.64 MMP9 (0.64) SLC1A3SLC1A2SLC1A1MMP13MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013010573-A1 COMPOUNDS WITH MATRIX-METALLOPROTEINASE INHIBITORY ACTIVITY UNIVERSITAET MUENSTER (DE) 2013-01-24 WO disclosed