SCHEMBL14764682

SCHEMBL14764682

O=C(O)c1cncc(Br)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.45
KDM4E B2RXH2 5/20 0.45
NAPRT Q6XQN6 1/20 0.45
ALDH1A1 P00352 4/20 0.42
POLB P06746 1/20 0.42
ALOX15 P16050 3/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TSHR P16473 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
ACMSD Q8TDX5 1/20 0.39
HIF1A Q16665 1/20 0.38
LMNA P02545 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
P4HA1 P13674 1/20 0.34
MIF P14174 1/20 0.34
P4HTM Q9NXG6 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
MC4R P32245 1/20 0.34
ADRA1A P35348 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL69399 0.83 KDM4E (0.55) HCAR2KDM4ENAPRTALDH1A1POLB
SCHEMBL13837305 0.80 ADORA3 (0.47) HCAR2KDM4EPOLBTSHRLMNA
SCHEMBL17449406 0.80 ALDH1A1 (0.33) HCAR2KDM4ENAPRTALDH1A1POLB
SCHEMBL31118151 0.79 HCAR2 (0.46) HCAR2KDM4ENAPRTALDH1A1POLB
SCHEMBL162262 0.79 HCAR2 (0.46) HCAR2KDM4ENAPRTALDH1A1POLB
Hydrochloric Acid SCHEMBL21752450 0.78 ADORA3 (0.45) HCAR2KDM4EPOLBTSHRLMNA
SCHEMBL29497681 0.77 HCAR2 (0.45) HCAR2KDM4ENAPRTALDH1A1POLB
SCHEMBL9478482 0.77 HCAR2 (0.45) HCAR2KDM4ENAPRTALDH1A1POLB
SCHEMBL17440722 0.75 MRGPRX4 (0.43) KDM4EALDH1A1SMN1; SMN2
SCHEMBL28139894 0.75 KDM4E (0.49) KDM4EALDH1A1HPGDLMNAADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747247-A1 NOVEL FATTY ACID AMIDE HYDROLASE MODULATORS, COMPOSITIONS COMPRISING THE SAME AND USES THEREOF Apogee Pharmaceuticals, Inc. (CA) 2026-05-27 EP disclosed
US-20250382283-A1 COMPOUNDS AND THEIR USES AS CD38 INHIBITORS NANJING IMMUNOPHAGE BIOTECH CO LTD (CN) 2025-12-18 US disclosed
WO-2025215110-A1 NEW AMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS SOS1 INHIBITORS LES LABORATOIRES SERVIER (FR) 2025-10-16 WO disclosed
US-12410137-B2 Fatty acid amide hydrolase modulators, compositions comprising the same and uses thereof APOGEE PHARMACEUTICALS, INC. (CA) 2025-09-09 US disclosed
US-20250197376-A1 PYRAZINE AMIDE DERIVATIVES NOVARTIS AG (CH) 2025-06-19 US disclosed
US-20250129027-A1 FATTY ACID AMIDE HYDROLASE MODULATORS, COMPOSITIONS COMPRISING THE SAME AND USES THEREOF APOGEE PHARMACEUTICALS, INC. (CA) 2025-04-24 US disclosed
EP-4499631-A1 PYRAZINE AMIDE DERIVATIVES Novartis AG (CH) 2025-02-05 EP disclosed
WO-2025015420-A1 NOVEL FATTY ACID AMIDE HYDROLASE MODULATORS, COMPOSITIONS COMPRISING THE SAME AND USES THEREOF APOGEE PHARMACEUTICALS, INC. (CA) 2025-01-23 WO disclosed
CN-118591538-A Pyrazinamide derivatives 诺华股份有限公司 2024-09-03 CN disclosed
US-20240254113-A1 COMPOUNDS AND THEIR USES AS CD38 INHIBITORS Nanjing Immunophage Biotech Co., Ltd. (CN) 2024-08-01 US disclosed
EP-3402799-B1 HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS ENANTA PHARM INC (US) 2022-05-04 EP disclosed
WO-2020030925-A1 HETEROCYCLIC SUBSTITUTED UREAS, FOR USE AGAINST CANCER ARTIOS PHARMA LIMITED (GB) 2020-02-13 WO disclosed
WO-2020030925-A1 HETEROCYCLIC SUBSTITUTED UREAS, FOR USE AGAINST CANCER ARTIOS PHARMA LIMITED (GB) 2020-02-13 WO disclosed
EP-3402799-A1 HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS Enanta Pharmaceuticals, Inc. (US) 2018-11-21 EP disclosed
EP-2753618-B1 HETEROCYCLIC-SUBSTITUED BENZOFURAN DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME (US) 2018-04-11 EP disclosed
US-20170226129-A1 HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS ENANTA PHARMACEUTICALS, INC. 2017-08-10 US disclosed
WO-2017123884-A1 HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2017-07-20 WO disclosed
US-9549917-B2 Heterocyclic-substituted benzofuran derivatives and methods of use thereof for the treatment of viral diseases MERCK SHARP & DOHME CORP. (US) 2017-01-24 US disclosed
US-20140199263-A1 HETEROCYCLIC-SUBSTITUTED BENZOFURAN DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME LLC 2014-07-17 US disclosed
WO-2013034047-A1 HETEROCYCLIC-SUBSTITUED BENZOFURAN DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME CORP. (US) 2013-03-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170226129-A1 HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS SIRT1, FURIN, SIRT5 HCAR2 387/4885KDM4E 1342/4885NAPRT 78/4885
US-20250129027-A1 FATTY ACID AMIDE HYDROLASE MODULATORS, COMPOSITIONS COMPRISING THE SAME AND USES THEREOF FAAH, FAAH2, MGLL HCAR2 64/4885KDM4E 1807/4885NAPRT 499/4885
US-12410137-B2 Fatty acid amide hydrolase modulators, compositions comprising the same and uses thereof FAAH, FAAH2, MGLL HCAR2 64/4885KDM4E 1807/4885NAPRT 499/4885
US-20250197376-A1 PYRAZINE AMIDE DERIVATIVES SIRT5, GLS2, ARG2 HCAR2 911/4885KDM4E 1301/4885NAPRT 954/4885
US-20140199263-A1 HETEROCYCLIC-SUBSTITUTED BENZOFURAN DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES HCCS, GTF3C5, EIF5B HCAR2 3549/4885KDM4E 2235/4885NAPRT 153/4885
US-20240254113-A1 COMPOUNDS AND THEIR USES AS CD38 INHIBITORS CD38, CD22, BCL6B HCAR2 980/4885KDM4E 2706/4885NAPRT 251/4885
US-20250382283-A1 COMPOUNDS AND THEIR USES AS CD38 INHIBITORS CD38, FCGRT, CD22 HCAR2 621/4885KDM4E 1675/4885NAPRT 374/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.