SCHEMBL1476907

SCHEMBL1476907

CC(C)(C)OC(=O)N1CCC(C#N)(CO)CC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CTSK P43235 1/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
NR1H2 P55055 1/20 0.40
HPGD P15428 1/20 0.39
EPHX2 P34913 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
ATM Q13315 1/20 0.39
JAK2 O60674 2/20 0.39
JAK1 P23458 2/20 0.39
GPR119 Q8TDV5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31451925 0.91 CTSK (0.42) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL2798365 0.88 USP2 (0.43) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL23071129 0.88 USP2 (0.45) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL17830842 0.88 USP2 (0.45) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL10529377 0.87 USP2 (0.44) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL20571615 0.87 USP2 (0.44) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL17176669 0.87 JAK2 (0.44) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL23283111 0.87 USP2 (0.44) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL21325460 0.86 CYP4F2 (0.43) USP2SMN1; SMN2CTSKMEN1KMT2A
SCHEMBL28709409 0.85 USP2 (0.43) USP2SMN1; SMN2CTSKMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 120 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4652159-A1 INHIBITORS OF KIF18A AND USES THEREOF Insilico Medicine IP Limited (HK) 2025-11-26 EP disclosed
US-20250340569-A1 INHIBITORS OF KIF18A AND USES THEREOF INSILICO MEDICINE IP LTD (CN) 2025-11-06 US disclosed
US-12441704-B2 Compounds active towards nuclear receptors NUEVOLUTION A/S (DK) 2025-10-14 US disclosed
EP-4620533-A2 ANTAGONIST COMPOUNDS Adorx therapeutics Limited (GB) 2025-09-24 EP disclosed
US-20250206745-A1 PYRROLOPYRIDAZINE DERIVATIVES AND RELATED USES NODTHERA LTD (GB) 2025-06-26 US disclosed
WO-2025124415-A1 TETRACYCLIC DERIVATIVES AS K-Ras G12D INHIBITORS NIKANG THERAPEUTICS INC. (US) 2025-06-19 WO disclosed
WO-2025123318-A1 TETRACYCLIC DERIVATIVES AS K-Ras G12D INHIBITORS SHANGHAI BLUERAY BIOPHARMA CO., LTD. (CN) 2025-06-19 WO disclosed
EP-4188924-B1 ANTAGONIST COMPOUNDS ADORX THERAPEUTICS LTD (GB) 2025-06-18 EP disclosed
EP-3340988-B1 ION CHANNEL INHIBITORY COMPOUNDS, PHARMACEUTICAL FORMULATIONS AND USES AFASCI INC (US) 2025-04-09 EP disclosed
WO-2025051241-A1 MACROCYCLIC COMPOUND AND ANTIBODY-DRUG CONJUGATE THEREOF 劲方医药科技(上海)股份有限公司 2025-03-13 WO disclosed
US-7915274-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-03-29 US disclosed
US-20090156575-A1 NOVEL DIAZASPIROALKANES AND THEIR USE FOR TREATMENT OF CCR8 MEDIATED DISEASES ASTRAZENECA AB (SE) 2009-06-18 US disclosed
US-20070293496-A1 Nitrogen containing heterocyclic compounds and medicines containing the same OZAKI FUMIHIRO 2007-12-20 US disclosed
US-7265108-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI CO., LTD. (JP) 2007-09-04 US disclosed
EP-1484327-B1 NITROGENOUS HETEROCYCLIC COMPOUND AND MEDICINE THEREOF EISAI R&D MAN CO LTD (JP) 2007-08-01 EP disclosed
WO-2007030061-A1 NOVEL DIAZASPIROALKANES AND THEIR USE FOR TREATMENT OF CCR8 MEDIATED DISEASES ASTRAZENECA AB (SE) 2007-03-15 WO disclosed
US-6995144-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI CO., LTD. (JP) 2006-02-07 US disclosed
US-20050245527-A1 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI R&D MANAGEMENT CO., LTD. (JP) 2005-11-03 US disclosed
EP-1484327-A1 NITROGENOUS HETEROCYCLIC COMPOUND AND MEDICINE THEREOF Eisai Co., Ltd. (JP) 2004-12-08 EP disclosed
US-20040167224-A1 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI R&D MANAGEMENT CO., LTD. (JP) 2004-08-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070293496-A1 Nitrogen containing heterocyclic compounds and medicines containing the same XDH, NQO1, CYP1A1 USP2 3639/4885SMN1; SMN2 1451/4885CTSK 3787/4885
US-20250340569-A1 INHIBITORS OF KIF18A AND USES THEREOF KIF18A, KIF18B, KIF2C USP2 1987/4885SMN1; SMN2 81/4885CTSK 1717/4885
US-20250206745-A1 PYRROLOPYRIDAZINE DERIVATIVES AND RELATED USES IL1B, NLRP3, NLRP1 USP2 2631/4885SMN1; SMN2 4456/4885CTSK 1823/4885
US-20090156575-A1 NOVEL DIAZASPIROALKANES AND THEIR USE FOR TREATMENT OF CCR8 MEDIATED DISEASES CCR8, CCR1, CCR10 USP2 1086/4885SMN1; SMN2 609/4885CTSK 4376/4885
US-12441704-B2 Compounds active towards nuclear receptors NCOA1, NR1H2, NCOA3 USP2 4401/4885SMN1; SMN2 4320/4885CTSK 3288/4885
US-20040167224-A1 Nitrogen containing heterocyclic compounds and medicines containing the same NQO1, CBR1, NOX1 USP2 3522/4885SMN1; SMN2 1325/4885CTSK 4257/4885
US-20050245527-A1 Nitrogen containing heterocyclic compounds and medicines containing the same XDH, NQO1, CYP1A1 USP2 3639/4885SMN1; SMN2 1451/4885CTSK 3787/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.