SCHEMBL14965417

SCHEMBL14965417

O=C(CN1CCOc2nc([N+](=O)[O-])cn2CC1)N1CCC(c2ccccc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.43
LMNA P02545 2/20 0.41
PARP1 P09874 1/20 0.40
KMT2A Q03164 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 5/20 0.38
THRA P10827 1/20 0.38
VDR P11473 1/20 0.38
THRB P10828 1/20 0.38
TERT O14746 1/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 3/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
POLB P06746 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TLR9 Q9NR96 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966005 0.84 PKM (0.45) LMNAKMT2ATDP1ALDH1A1GAA
SCHEMBL14965582 0.80 HSD17B10 (0.38) LMNAKMT2ATDP1ALDH1A1MAPT
SCHEMBL14965808 0.79 LMNA (0.47) LMNAKMT2ATDP1ALDH1A1MAPT
SCHEMBL14965604 0.77 THRB (0.34) LMNATDP1ALDH1A1THRBGAA
SCHEMBL14966123 0.76 KMT2A (0.52) NAMPTLMNAKMT2ATDP1ALDH1A1
SCHEMBL14965773 0.76 L3MBTL1 (0.46) LMNAKMT2ATDP1ALDH1A1GAA
SCHEMBL14965756 0.76 PKM (0.40) LMNAALDH1A1SMN1; SMN2POLBKDM4E
SCHEMBL14965791 0.74 KDM4E (0.36) LMNAKMT2ATDP1ALDH1A1POLB
SCHEMBL14966168 0.74 ALDH1A1 (0.40) LMNAKMT2AALDH1A1SMN1; SMN2POLB
SCHEMBL14965832 0.74 NPC1 (0.36) LMNAKMT2AALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed