SCHEMBL15469468

SCHEMBL15469468

O=C1CCOc2ccc(Cl)nc21

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.38
MAOA P21397 1/20 0.38
MAP3K14 Q99558 1/20 0.35
GRM5 P41594 6/20 0.33
DYRK1A Q13627 3/20 0.32
DYRK2 Q92630 2/20 0.31
DYRK1B Q9Y463 2/20 0.31
TDP2 O95551 1/20 0.31
NSD2 O96028 1/20 0.31
NPC1 O15118 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10286589 0.79 S100A4 (0.38) MAOBMAOAMAP3K14GRM5DYRK1A
SCHEMBL15469476 0.79 MAOB (0.38) MAOBMAOAMAP3K14GRM5DYRK1A
SCHEMBL23376851 0.79 MAOB (0.38) MAOBMAOAMAP3K14GRM5DYRK1A
SCHEMBL23376935 0.79 MAOB (0.41) MAOBMAOAMAP3K14GRM5DYRK1A
SCHEMBL15469486 0.75 MAPT (0.37) MAOBMAOAMAP3K14GRM5DYRK1A
SCHEMBL25522617 0.75 MAOA (0.35) MAOBMAOAMAP3K14GRM5
SCHEMBL21935993 0.73 DYRK1A (0.35) DYRK1ANPC1POLBMAPTRAB9A
SCHEMBL1516800 0.72 MAP3K14 (0.40) MAP3K14DYRK1ADYRK1BMAPTRAB9A
SCHEMBL25832196 0.72 GRM5 (0.34) GRM5TDP2NSD2MAPT
SCHEMBL22439215 0.71 GRM5 (0.52) MAOBMAOAGRM5TDP2NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230002426-A1 CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL RECURIUM IP HOLDINGS, LLC 2023-01-05 US disclosed
WO-2021097139-A1 CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL RECURIUM IP HOLDINGS, LLC (US) 2021-05-20 WO disclosed
US-8952009-B2 Chroman derivatives as TRPM8 inhibitors AMGEN INC. (US) 2015-02-10 US disclosed
US-8952009-B2 Chroman derivatives as TRPM8 inhibitors AMGEN INC. (US) 2015-02-10 US disclosed
US-20140045855-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS AMGEN INC. (US) 2014-02-13 US disclosed
US-20140045855-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS AMGEN INC. (US) 2014-02-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140045855-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS TRPM8, TRPM5, TRPM7 MAOB 1631/4885MAOA 601/4885MAP3K14 1097/4885
US-20230002426-A1 CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL ADH1A, ADH1C, ADH5 MAOB 1691/4885MAOA 2803/4885MAP3K14 755/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.