SCHEMBL15469486

SCHEMBL15469486

COc1ccc2c(n1)C(=O)CCO2

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
LMNA P02545 1/20 0.37
SCN9A Q15858 3/20 0.36
GRM5 P41594 1/20 0.35
MAOB P27338 2/20 0.35
MAOA P21397 1/20 0.35
TXNRD1 Q16881 2/20 0.34
MAP3K14 Q99558 1/20 0.33
OGA O60502 1/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
BTK Q06187 1/20 0.32
DYRK1A Q13627 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
NNMT P40261 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23376851 0.78 MAOB (0.38) MAPTLMNAGRM5MAOBMAOA
SCHEMBL10286589 0.78 S100A4 (0.38) MAPTGRM5MAOBMAOAMAP3K14
SCHEMBL15469468 0.75 MAOB (0.38) MAPTGRM5MAOBMAOAMAP3K14
SCHEMBL23376935 0.75 MAOB (0.41) GRM5MAOBMAOAMAP3K14DYRK1A
SCHEMBL15469476 0.75 MAOB (0.38) MAPTGRM5MAOBMAOAMAP3K14
SCHEMBL18237885 0.74 MAOA (0.35) GRM5MAOBMAOAMAP3K14MTNR1B
SCHEMBL25522617 0.74 MAOA (0.35) GRM5MAOBMAOAMAP3K14
SCHEMBL23376843 0.73 MEN1 (0.37) POLBTDP1NNMTMTNR1AMTNR1B
SCHEMBL874647 0.70 ALDH1A1 (0.37) MAPTLMNAMAOBMAOAPOLB
SCHEMBL10286843 0.67 MAOB (0.37) GRM5MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230002426-A1 CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL RECURIUM IP HOLDINGS, LLC 2023-01-05 US disclosed
WO-2021097139-A1 CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL RECURIUM IP HOLDINGS, LLC (US) 2021-05-20 WO disclosed
US-8952009-B2 Chroman derivatives as TRPM8 inhibitors AMGEN INC. (US) 2015-02-10 US disclosed
US-8952009-B2 Chroman derivatives as TRPM8 inhibitors AMGEN INC. (US) 2015-02-10 US disclosed
US-20150031668-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS AMGEN INC (US) 2015-01-29 US disclosed
US-20150031668-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS AMGEN INC (US) 2015-01-29 US disclosed
US-20140045855-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS AMGEN INC. (US) 2014-02-13 US disclosed
US-20140045855-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS AMGEN INC. (US) 2014-02-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150031668-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS TRPM8, TRPM5, TRPM7 MAPT 727/4885LMNA 710/4885SCN9A 66/4885
US-20140045855-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS TRPM8, TRPM5, TRPM7 MAPT 727/4885LMNA 710/4885SCN9A 66/4885
US-20230002426-A1 CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL ADH1A, ADH1C, ADH5 MAPT 2641/4885LMNA 900/4885SCN9A 4013/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.