SCHEMBL15534816

SCHEMBL15534816

COC(=O)C1CCCCC1CNC(=O)c1c(N)cccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.47
SLC6A9 P48067 10/20 0.41
TAS1R3 Q7RTX0 2/20 0.40
TAS1R1 Q7RTX1 2/20 0.40
JAK1 P23458 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
DRD2 P14416 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR4 Q13639 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
DPP4 P27487 1/20 0.38
PREP P48147 1/20 0.38
FAP Q12884 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15535647 0.87 DRD2 (0.47) TAS1R3TAS1R1DRD2HTR3EHTR3B
SCHEMBL15534876 0.82 DRD2 (0.38) TAS1R3TAS1R1DRD2HTR3EHTR3B
SCHEMBL1666992 0.81 ALDH1A1 (0.46) DRD2HTR3EHTR3BHTR3AHTR4
SCHEMBL1666286 0.71 SLC6A2 (0.40) DPP4
SCHEMBL22447716 0.71 DRD2 (0.44) DRD2HTR3EHTR3BHTR3AHTR4
SCHEMBL8932345 0.71 P2RX7 (0.57) P2RX7SLC6A9JAK1
SCHEMBL9017627 0.70 MAPK14 (0.55) P2RX7TAS1R3TAS1R1JAK1TAS1R2
SCHEMBL1668136 0.69 HPGD (0.50)
SCHEMBL8732695 0.69 P2RX7 (0.58) P2RX7SLC6A9JAK1
SCHEMBL15534872 0.68 CCNA2 (0.45) PREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013177349-A2 QUINAZOLINEDIONES AS TANKYRASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-11-28 WO disclosed