SCHEMBL15535647

SCHEMBL15535647

COC(=O)C1CCCCC1CNC(=O)c1c(N)cccc1OC

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.47
POLB P06746 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
ADORA2A P29274 1/20 0.38
HPGD P15428 2/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR4 Q13639 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
RCE1 Q9Y256 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15534816 0.87 P2RX7 (0.47) DRD2TAS1R3TAS1R1HTR3EHTR3B
SCHEMBL15534876 0.82 DRD2 (0.38) DRD2TAS1R3TAS1R1L3MBTL1HPGD
SCHEMBL1666992 0.81 ALDH1A1 (0.46) DRD2HPGDHTR3EHTR3BHTR3A
SCHEMBL1666286 0.71 SLC6A2 (0.40) TAAR1HPGDKDM4EALDH1A1
SCHEMBL22447716 0.71 DRD2 (0.44) DRD2POLBHPGDHTR3EHTR3B
SCHEMBL2241114 0.70 HPGD (0.63) POLBL3MBTL1TAAR1HPGDKDM4E
SCHEMBL1558671 0.69 CA12 (0.52) POLBTAAR1HPGDKDM4EALDH1A1
SCHEMBL1558070 0.69 CA12 (0.52) POLBTAAR1HPGDKDM4EALDH1A1
SCHEMBL1668136 0.69 HPGD (0.50) L3MBTL1HPGDKDM4EALDH1A1
SCHEMBL12986205 0.69 AAK1 (0.41) TAS1R3TAS1R1HTR4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013177349-A2 QUINAZOLINEDIONES AS TANKYRASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-11-28 WO disclosed