SCHEMBL16150671

SCHEMBL16150671

COc1c(C(=O)Nc2c(Br)cc(C(F)(C(F)(F)F)C(F)(F)F)cc2OC(F)F)cccc1N(C)C(=O)c1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 17/20 0.38
MLYCD O95822 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29376079 1.00 GPBAR1 (0.38) GPBAR1MLYCDRXFP1ALDH1A1MAPT
SCHEMBL21574048 0.92 GPBAR1 (0.36) GPBAR1MLYCDRXFP1ALDH1A1MAPT
SCHEMBL22332345 0.92 GPBAR1 (0.38) GPBAR1MLYCDRXFP1ALDH1A1MAPT
SCHEMBL14844306 0.91 GPBAR1 (0.40) GPBAR1MLYCDRXFP1ALDH1A1MAPT
SCHEMBL16868757 0.91 GPBAR1 (0.36) GPBAR1MLYCDRXFP1
SCHEMBL18354632 0.91 MLYCD (0.36) GPBAR1MLYCDRXFP1ALDH1A1MAPT
SCHEMBL16863570 0.90 PDE4A (0.33) GPBAR1RXFP1ALDH1A1MAPTSMN1; SMN2
SCHEMBL18355489 0.88 MLYCD (0.35) GPBAR1MLYCDALDH1A1MAPTHTT
SCHEMBL16863611 0.87 MLYCD (0.34) MLYCDALDH1A1MAPTHTTSMN1; SMN2
SCHEMBL18359968 0.86 RXFP1 (0.42) RXFP1ALDH1A1HTTSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 117 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260047580-A1 HETEROCYCLIC COMPOUND AND HARMFUL ARTHROPOD PEST CONTROL COMPOSITION CONTAINING SAME SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2026-02-19 US disclosed
US-12478067-B2 Heterocyclic compound and harmful arthropod pest control composition containing same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2025-11-25 US disclosed
EP-3778583-B1 HETEROCYCLIC COMPOUND AND ARTHROPOD PEST CONTROL COMPOSITION CONTAINING SAME SUMITOMO CHEMICAL CO (JP) 2025-06-18 EP disclosed
US-12234247-B2 Heterocyclic compound and harmful arthropod-controlling composition containing same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2025-02-25 US disclosed
US-12225904-B2 Phenylpyrazole compound and method for controlling plant disease SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2025-02-18 US disclosed
US-12221431-B2 Heterocyclic compound SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2025-02-11 US disclosed
US-12172978-B2 Ether compound and harmful arthropod-controlling composition containing same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2024-12-24 US disclosed
US-20240389582-A1 ACRYLATE DERIVATIVE, USE AND PRODUCTION INTERMEDIATE COMPOUND OF THE SAME SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2024-11-28 US disclosed
US-20240389583-A1 ACRYLATE DERIVATIVE, USE AND PRODUCTION INTERMEDIATE COMPOUND OF THE SAME SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2024-11-28 US disclosed
EP-3918896-B1 HETEROCYCLIC COMPOUND AND HARMFUL ARTHROPOD CONTROL COMPOSITION CONTAINING SAME SUMITOMO CHEMICAL CO (JP) 2024-11-27 EP disclosed
US-20170000121-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2017-01-05 US disclosed
EP-3087052-A1 INSECTICIDAL COMPOUNDS Syngenta Participations AG (CH) 2016-11-02 EP disclosed
EP-3087053-A1 INSECTICIDAL COMPOUNDS Syngenta Participations AG (CH) 2016-11-02 EP disclosed
US-20160168097-A1 PROCESS FOR THE PREPARATION OF AMIDES FROM HINDERED ANILINES CONTAINING A PERHALOALKYL GROUP SYNGENTA PARTICIPATIONS AG (CH) 2016-06-16 US disclosed
US-20160168097-A1 PROCESS FOR THE PREPARATION OF AMIDES FROM HINDERED ANILINES CONTAINING A PERHALOALKYL GROUP SYNGENTA PARTICIPATIONS AG (CH) 2016-06-16 US disclosed
EP-2981519-A1 PROCESS FOR THE PREPARATION OF AMIDES FROM HINDERED ANILINES CONTAINING A PERHALOALKYL GROUP Syngenta Participations AG (CH) 2016-02-10 EP disclosed
WO-2015097091-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2015-07-02 WO disclosed
WO-2015097094-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2015-07-02 WO disclosed
WO-2014161850-A1 PROCESS FOR THE PREPARATION OF AMIDES FROM HINDERED ANILINES CONTAINING A PERHALOALKYL GROUP SYNGENTA PARTICIPATIONS AG (CH) 2014-10-09 WO disclosed
WO-2014161850-A1 PROCESS FOR THE PREPARATION OF AMIDES FROM HINDERED ANILINES CONTAINING A PERHALOALKYL GROUP SYNGENTA PARTICIPATIONS AG (CH) 2014-10-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12225904-B2 Phenylpyrazole compound and method for controlling plant disease HRH3, H1-3, HRH4 GPBAR1 1441/4885MLYCD 555/4885RXFP1 467/4885
US-20160168097-A1 PROCESS FOR THE PREPARATION OF AMIDES FROM HINDERED ANILINES CONTAINING A PERHALOALKYL GROUP ABHD5, FADS1, PFAS GPBAR1 1810/4885MLYCD 1591/4885RXFP1 3588/4885
US-20170000121-A1 INSECTICIDAL COMPOUNDS ACHE, NIT2, CHRM1 GPBAR1 1869/4885MLYCD 3166/4885RXFP1 1005/4885
US-20240389583-A1 ACRYLATE DERIVATIVE, USE AND PRODUCTION INTERMEDIATE COMPOUND OF THE SAME C1S, ACR, AKR1C3 GPBAR1 3532/4885MLYCD 364/4885RXFP1 3300/4885
US-12221431-B2 Heterocyclic compound NR4A2, NR4A1, NR2C2 GPBAR1 687/4885MLYCD 4561/4885RXFP1 622/4885
US-12478067-B2 Heterocyclic compound and harmful arthropod pest control composition containing same C5, COX6C, C1S GPBAR1 2548/4885MLYCD 1199/4885RXFP1 364/4885
US-20260047580-A1 HETEROCYCLIC COMPOUND AND HARMFUL ARTHROPOD PEST CONTROL COMPOSITION CONTAINING SAME COX6C, COX6B1, CYC1 GPBAR1 1987/4885MLYCD 1160/4885RXFP1 519/4885
US-20240389582-A1 ACRYLATE DERIVATIVE, USE AND PRODUCTION INTERMEDIATE COMPOUND OF THE SAME C1S, ACR, AKR1C3 GPBAR1 3532/4885MLYCD 364/4885RXFP1 3300/4885
US-12234247-B2 Heterocyclic compound and harmful arthropod-controlling composition containing same C5, COX6C, COX6B1 GPBAR1 3078/4885MLYCD 3926/4885RXFP1 521/4885
US-12172978-B2 Ether compound and harmful arthropod-controlling composition containing same C3AR1, C5, CYP1B1 GPBAR1 830/4885MLYCD 2839/4885RXFP1 602/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.