Cromitrile Sodium

Cromitrile Sodium

SCHEMBL1649767

N#Cc1ccc(OCC(O)COc2cccc3oc(-c4nn[n-]n4)cc(=O)c23)cc1.[Na+]

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Cromitrile Sodium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 2/20 0.46
HIF1A Q16665 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
LMNA P02545 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
AR P10275 2/20 0.40
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
MAOB P27338 6/20 0.35
MAOA P21397 4/20 0.35
HPGD P15428 2/20 0.34
TNKS O95271 1/20 0.34
AGER Q15109 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
ALDH1A1 P00352 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cromitrile Sodium SCHEMBL636215 0.84 GPR35 (0.46) GPR35HIF1AMEN1KMT2ALMNA
Cromitrile SCHEMBL11475038 0.80 GPR35 (0.46) GPR35HIF1AMEN1KMT2ALMNA
Cromitrile SCHEMBL11480432 0.79 GPR35 (0.46) GPR35HIF1AMEN1KMT2ALMNA
Cromitrile SCHEMBL11480428 0.79 GPR35 (0.46) GPR35HIF1AMEN1KMT2ALMNA
SCHEMBL11482479 0.79 GPR35 (0.57) GPR35HIF1AMEN1KMT2ALMNA
SCHEMBL11478244 0.77 GPR35 (0.78) GPR35HIF1AMEN1KMT2ALMNA
SCHEMBL11348725 0.77 GPR35 (0.78) GPR35HIF1AMEN1KMT2ALMNA
SCHEMBL11478258 0.76 GPR35 (0.76) GPR35HIF1AMEN1KMT2ALMNA
SCHEMBL11478579 0.73 GPR35 (0.59) GPR35HIF1AMEN1KMT2ALMNA
SCHEMBL11657040 0.72 GPR35 (0.62) GPR35HIF1AMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7927613-B2 Pharmaceutical co-crystal compositions UNIVERSITY OF SOUTH FLORIDA (US) 2011-04-19 US disclosed
US-7790905-B2 Pharmaceutical propylene glycol solvate compositions MCNEIL-PPC, INC. (US) 2010-09-07 US disclosed