Arsanilic Acid

Arsanilic Acid

SCHEMBL1649934

Nc1ccc([As](=O)([O-])O)cc1.[Na+]

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Arsanilic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB known ✓ P10828 1/20 0.36
CA4 known ✓ P22748 2/20 0.36
CA1 known ✓ P00915 2/20 0.36
CA2 known ✓ P00918 2/20 0.36
CA12 known ✓ O43570 1/20 0.36
TSHR P16473 4/20 0.62
KDM4E B2RXH2 2/20 0.62
RAB9A P51151 2/20 0.62
ALDH1A1 P00352 6/20 0.39
NT5E P21589 1/20 0.39
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP3A4 P08684 3/20 0.37
LMNA P02545 2/20 0.37
CYP2C9 P11712 2/20 0.37
MPO P05164 1/20 0.37
HTR6 P50406 1/20 0.37
TDP1 Q9NUW8 4/20 0.36
TDP2 O95551 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL886902 0.88 CYP2C19 (0.53) TSHRKDM4ERAB9AALDH1A1NT5E
Arsanilic Acid SCHEMBL31473000 0.80 CA4 (0.56) TSHRKDM4ERAB9AALDH1A1NT5E
Arsanilic Acid SCHEMBL4837583 0.77 KDM4E (1.00) TSHRKDM4ERAB9AALDH1A1NT5E
Arsanilic Acid SCHEMBL160507 0.77 KDM4E (1.00) TSHRKDM4ERAB9AALDH1A1NT5E
SCHEMBL28056036 0.76 TSHR (0.68) TSHRKDM4ERAB9AALDH1A1NT5E
Arsanilic Acid SCHEMBL5051668 0.75 KDM4E (0.95) TSHRKDM4ERAB9AALDH1A1NT5E
Arsanilic Acid SCHEMBL31473003 0.75 TSHR (0.95) TSHRKDM4ERAB9AALDH1A1NT5E
SCHEMBL4407102 0.71 TSHR (0.45) TSHRKDM4ERAB9AALDH1A1NT5E
Difetarsone SCHEMBL5058528 0.70 ALDH1A1 (0.43) ALDH1A1MAPTMEN1KMT2ALMNA
Difetarsone SCHEMBL160476 0.70 ALDH1A1 (0.43) ALDH1A1MAPTMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2744790-B1 FUNGICIDAL SUBSTITUTED 1-{2-[2-HALO-4-(4-HALOGEN-PHENOXY)-PHENYL]-2-ALKOXY-2-ALKYNYL/ALKENYL-ETHYL}-1H-[1,2,4]TRIAZOLE COMPOUNDS BASF SE (DE) 2016-04-27 EP claimed
CN-101214397-A Medicament elution bracket for promoting esoderma repair and preventing vascular restenosis WEI YANG (CN) 2008-07-09 CN claimed
EP-1757607-A1 N5-substituted benzo¬2,3|azepino¬4,5-b|indol-6-ones for treating tropical diseases Molisa GmbH (DE) 2007-02-28 EP claimed
US-20250387364-A1 ARSINOTHRICIN AND METHODS OF TREATING INFECTIONS USING ARSINOTHRICIN THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2025-12-25 US disclosed
EP-4664445-A1 PHYSICAL COMPRESSION DEVICE WITH ARTIFICIAL INTELLIGENCE ASSISTANCE, ON A SYMBOL STAGE, EQUIVALENT PROJECTION OF SEVERAL LEVELS OF ARRANGEMENT BY VIRTUAL PIANO Valéry-Daulon, Marc (FR) 2025-12-17 EP disclosed
US-12414932-B2 Arsinothricin and methods of treating infections using arsinothricin THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2025-09-16 US disclosed
US-20250241885-A1 ARSINOTHRICIN AND METHODS OF TREATING INFECTIONS USING ARSINOTHRICIN THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2025-07-31 US disclosed
US-12303485-B2 Arsinothricin and methods of treating infections using arsinothricin THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2025-05-20 US disclosed
CN-119776293-A ArsL mutant and application thereof in synthesis of Arsinothricin 上海交通大学 2025-04-08 CN disclosed
WO-2024232889-A1 ENHANCING BOREHOLE RESONANCE SIGNAL FOR THROUGH TUBING CEMENT EVALUATION HALLIBURTON ENERGY SERVICES, INC. (US) 2024-11-14 WO disclosed
US-12134695-B2 Aqueous binder formulation based on functionalized polyurethanes BASF SE (DE) 2024-11-05 US disclosed
EP-0185393-A1 Process for decontaminating the surface of an object Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 1986-06-25 EP disclosed
US-4569836-A Cancer treatment by intracellular hyperthermia GORDON, DAVID, SKOKIE, ILLINOIS 1986-02-11 US disclosed
US-4554959-A Surface treatment of sheet material RY AB, FACK (SE) 1985-11-26 US disclosed
EP-0002596-B1 METHOD FOR REDUCING THE AMOUNT OF FREE FORMALDEHYDE IN AN AMINO FORMALDEHYDE RESIN BEROL KEMI AB (SE) 1983-07-27 EP disclosed
US-4359453-A Atherosclerosis treatment method GORDON, DAVID, SKOKIE, ILLINOIS 1982-11-16 US disclosed
US-4303636-A Cancer treatment GORDON, DAVID, SKOKIE, ILLINOIS 1981-12-01 US disclosed
EP-0002596-A1 Method for reducing the amount of free formaldehyde in an amino formaldehyde resin BEROL KEMI AB (SE) 1979-06-27 EP disclosed
EP-0001485-A2 Herbicidal sulphonamides, their preparation, compositions containing them and use thereof E.I. DU PONT DE NEMOURS AND COMPANY (US) 1979-04-18 EP disclosed
US-4106488-A Cancer treatment method GORDON, DAVID, SKOKIE, ILLINOIS 1978-08-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250387364-A1 ARSINOTHRICIN AND METHODS OF TREATING INFECTIONS USING ARSINOTHRICIN ARSA, NAT1, NAA15 THRB 343/4885CA4 3529/4885CA1 3261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.