Senazodan

Senazodan

SCHEMBL1652002

O=C1CCC(c2ccc(Nc3ccncc3)cc2)=NN1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 1.00
PDE3B Q13370 13/20 0.57
PDE3A Q14432 12/20 0.57
PDE4A P27815 4/20 0.57
PDE4B Q07343 4/20 0.57
PDE4C Q08493 4/20 0.57
PDE4D Q08499 4/20 0.57
LMNA P02545 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
TSHR P16473 1/20 0.57
MAPK1 P28482 1/20 0.57
CYP2C19 P33261 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
MAPT P10636 2/20 0.48
NPY1R P25929 1/20 0.48
NPY2R P49146 1/20 0.48
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Senazodan SCHEMBL4519202 0.98 KCNH2 (0.97) KCNH2PDE3BPDE3APDE4APDE4B
Senazodan SCHEMBL1649599 0.98 KCNH2 (0.97) KCNH2PDE3BPDE3APDE4APDE4B
Senazodan SCHEMBL4526209 0.97 KCNH2 (0.94) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL7263634 0.85 KCNH2 (0.73) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL10548193 0.84 KCNH2 (0.71) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL7264027 0.82 KCNH2 (0.70) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL10353452 0.82 SMN1; SMN2 (0.81) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL10474131 0.81 KCNH2 (0.67) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL22910067 0.80 KCNH2 (0.66) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL2478615 0.80 KCNH2 (0.66) KCNH2PDE3BPDE3APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090062295-A1 Pharmaceutical Products MITSUBISHI PHARMA CORPORATION (JP) 2009-03-05 US claimed
EP-1864664-A1 PHARMACEUTICAL PREPARATION Mitsubishi Pharma Corporation (JP) 2007-12-12 EP claimed
US-6110471-A ADMINISTERING PHOSPHODIESTERASE FOR INHIBITION OF THE CYCLES THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2000-08-29 US claimed
US-4971968-A CARDIOVASCULAR DISORDERS, STIMULANTS MITSUBISHI KASEI CORPORATION (JP) 1990-11-20 US claimed
EP-0145019-A2 Pyridazinone derivatives and salts thereof MITSUBISHI KASEI CORPORATION (JP) 1985-06-19 EP claimed
JP-60126282-A None JP disclosed
US-12472186-B2 Pharmaceutical compositions and methods of treating cardiovascular diseases Cardix Therapeutics LLC (US) 2025-11-18 US disclosed
US-20250345308-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING CONDITIONS ANSELLA THERAPEUTICS INC (US) 2025-11-13 US disclosed
US-12201607-B2 Compositions and methods for preventing and treating conditions Ansella Therapeutics, Inc. (US) 2025-01-21 US disclosed
US-20240285639-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2024-08-29 US disclosed
US-20240207279-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2024-06-27 US disclosed
US-11951107-B2 Deuterated pharmaceutical compositions and methods of treating cardiovascular diseases CARDIX Therapeutics, LLC (US) 2024-04-09 US disclosed
US-20040063710-A1 Ophthalmological preparations MITSUBISHI PHARMA CORPORATION (JP) 2004-04-01 US disclosed
EP-1400520-A1 CRYSTAL OF 6- 4-(4-PYRIDYLAMINO)PHENYL]-4, 5-DIHYDRO-3(2H)-PYRIDAZINONE HYDROCHLORIDE TRIHYDRATE Mitsubishi Pharma Corporation (JP) 2004-03-24 EP disclosed
EP-1346728-A1 OPHTHALMOLOGICAL PREPARATIONS Mitsubishi Pharma Corporation (JP) 2003-09-24 EP disclosed
WO-2002088109-A1 CRYSTAL OF 6-[4-(4-PYRIDYLAMINO)PHENYL]-4, 5-DIHYDRO-3(2H)-PYRIDAZINONE HYDROCHLORIDE TRIHYDRATE MITSUBISHI PHARMA CORPORATION (JP) 2002-11-07 WO disclosed
WO-2002088109-A1 CRYSTAL OF 6-[4-(4-PYRIDYLAMINO)PHENYL]-4, 5-DIHYDRO-3(2H)-PYRIDAZINONE HYDROCHLORIDE TRIHYDRATE MITSUBISHI PHARMA CORPORATION (JP) 2002-11-07 WO disclosed
US-4971968-A CARDIOVASCULAR DISORDERS, STIMULANTS MITSUBISHI KASEI CORPORATION (JP) 1990-11-20 US disclosed
JP-S60126282-A PYRIDAZINONE DERIVATIVE OF SALT THEREOF MITSUBISHI CHEM IND LTD 1985-07-05 JP disclosed
EP-0145019-A2 Pyridazinone derivatives and salts thereof MITSUBISHI KASEI CORPORATION (JP) 1985-06-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11951107-B2 Deuterated pharmaceutical compositions and methods of treating cardiovascular diseases ADRB2, ADRA2C, ADRB1 KCNH2 296/4885PDE3B 84/4885PDE3A 81/4885
US-20240285639-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES ADRB2, ADRA2C, ADRB1 KCNH2 296/4885PDE3B 84/4885PDE3A 81/4885
US-12201607-B2 Compositions and methods for preventing and treating conditions LIPA, COL2A1, COL1A1 KCNH2 3836/4885PDE3B 1086/4885PDE3A 638/4885
US-20090062295-A1 Pharmaceutical Products H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, DPP4, CYP2D6 KCNH2 768/4885PDE3B 207/4885PDE3A 130/4885
US-20040063710-A1 Ophthalmological preparations EYA3, AQP4, AQP3 KCNH2 52/4885PDE3B 406/4885PDE3A 117/4885
US-20250345308-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING CONDITIONS LIPA, COL2A1, COL1A1 KCNH2 3836/4885PDE3B 1086/4885PDE3A 638/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.