SCHEMBL16612679

SCHEMBL16612679

COc1ccc2c(CCn3c[c]c(C(N)=O)n3)c[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.52
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
MTNR1A P48039 3/20 0.51
MTNR1B P49286 2/20 0.51
HTR6 P50406 1/20 0.47
MAPT P10636 3/20 0.46
ADORA2A P29274 1/20 0.45
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
GAA P10253 1/20 0.43
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12479180 0.92 MTNR1A (0.55) HTR2AMEN1KMT2AMTNR1AMTNR1B
SCHEMBL16612878 0.82 KMT2A (0.46) HTR2AMEN1KMT2AHTR6MAPT
SCHEMBL16612770 0.81 ADRB2 (0.44) MEN1KMT2AMTNR1AMTNR1BHTR6
SCHEMBL16612796 0.79 ADRB2 (0.55) MEN1KMT2AMTNR1AMTNR1BHTR6
SCHEMBL16612788 0.78 MPO (0.56) HTR2AKMT2AMTNR1AMTNR1B
SCHEMBL16612934 0.78 HTR2A (0.52) HTR2AMTNR1AMTNR1BHTR6HCRTR2
SCHEMBL16612961 0.78 MTNR1A (0.53) MEN1KMT2AMTNR1AMTNR1BHTR6
SCHEMBL16612943 0.76 SIGMAR1 (0.47) MTNR1AMTNR1B
SCHEMBL8020879 0.73 HTR2A (0.67) HTR2AMEN1KMT2AMTNR1AMTNR1B
SCHEMBL16612680 0.72 HTR2A (0.58) HTR2AMEN1KMT2AMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed