SCHEMBL16612796

SCHEMBL16612796

COc1ccc2c(c1)c(CCn1c[c]c(C(N)=O)n1)cn2C

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.55
MTNR1A P48039 12/20 0.53
MTNR1B P49286 11/20 0.53
NQO2 P16083 1/20 0.53
HTR6 P50406 1/20 0.50
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612770 0.92 ADRB2 (0.44) ADRB2MTNR1AMTNR1BNQO2HTR6
SCHEMBL16612684 0.83 HTR2A (0.49) MEN1KMT2AALDH1A1LMNA
SCHEMBL12479180 0.81 MTNR1A (0.55) MTNR1AMTNR1BNQO2HTR6MEN1
SCHEMBL16612679 0.79 HTR2A (0.52) MTNR1AMTNR1BHTR6HCRTR1HCRTR2
SCHEMBL16612943 0.76 SIGMAR1 (0.47) MTNR1AMTNR1B
SCHEMBL16612868 0.76 MTNR1A (0.49) MTNR1AMTNR1BHCRTR1HCRTR2RAB9A
SCHEMBL16612854 0.73 MTNR1A (0.52) MTNR1AMTNR1BHCRTR1HCRTR2MEN1
SCHEMBL18509701 0.73 MTNR1A (0.67) ADRB2MTNR1AMTNR1BNQO2HTR6
SCHEMBL12479701 0.73 ADRB2 (0.63) ADRB2MTNR1AMTNR1BNQO2HTR6
SCHEMBL16612856 0.72 MTNR1A (0.54) MTNR1AMTNR1BHCRTR1HCRTR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed