SCHEMBL16659465

SCHEMBL16659465

CC1=NN(c2cccnc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.45
CYP2E1 P05181 2/20 0.45
CYP3A4 P08684 2/20 0.45
CHRNB2 P17787 3/20 0.42
CHRNA4 P43681 3/20 0.42
MAOB P27338 1/20 0.41
MAPT P10636 4/20 0.39
NPSR1 Q6W5P4 2/20 0.39
TSHR P16473 1/20 0.39
TDP1 Q9NUW8 2/20 0.39
HTT P42858 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
RECQL P46063 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
GLA P06280 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1122272 0.80 MAOB (0.59) CYP3A4CHRNB2CHRNA4MAOBMAPT
SCHEMBL16652173 0.79 ABL1 (0.44) CYP2A6CYP3A4CHRNB2CHRNA4MAPT
SCHEMBL10417191 0.79 ALOX5 (0.51) CYP2A6CYP3A4CHRNB2CHRNA4MAPT
SCHEMBL20284826 0.78 CHKA (0.42) MAOBMAPTNPSR1TSHRTDP1
SCHEMBL2731119 0.76 MAPT (0.73) CHRNB2CHRNA4MAOBMAPTTDP1
SCHEMBL13260410 0.72 MAOB (0.54) MAOBMAPTNPSR1TSHRTDP1
SCHEMBL31065089 0.69 MAOB (0.51) CYP3A4CHRNB2CHRNA4MAOBMAPT
SCHEMBL27681500 0.69 MAPT (0.73) CYP2A6CYP3A4MAOBMAPTTDP1
SCHEMBL31415059 0.68 ADRB1 (0.44) CYP3A4MAOBMAPTNPSR1TSHR
SCHEMBL30720445 0.68 CHRNB2 (0.45) CYP2A6CYP2E1CYP3A4CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170101392-A1 PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS DOW AGROSCIENCES LLC (US) 2017-04-13 US disclosed
US-9611247-B2 Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine DOW AGROSCIENCES LLC (US) 2017-04-04 US disclosed
US-20160031850-A1 PROCESS FOR THE PREPARATION OF 3-(3-CHLORO-1H-PYRAZOL-1-YL)PYRIDINE DOW AGROSCIENCES LLC 2016-02-04 US disclosed
US-9249122-B1 Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine DOW AGROSCIENCES LLC 2016-02-02 US disclosed
US-9199964-B1 Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine DOW AGROSCIENCES LLC (US) 2015-12-01 US disclosed
US-20150250177-A1 PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS DOW AGROSCIENCES LLC 2015-09-10 US disclosed
US-9108946-B2 Processes for the preparation of pesticidal compounds DOW AGROSCIENCES LLC (US) 2015-08-18 US disclosed
US-20150112078-A1 PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS DOW AGROSCIENCES LLC 2015-04-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150112078-A1 PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS DDT, ACHE, PTMS CYP2A6 457/4885CYP2E1 111/4885CYP3A4 98/4885
US-20170101392-A1 PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS DDT, ACHE, PTMS CYP2A6 457/4885CYP2E1 111/4885CYP3A4 98/4885
US-20160031850-A1 PROCESS FOR THE PREPARATION OF 3-(3-CHLORO-1H-PYRAZOL-1-YL)PYRIDINE PPOX, PDXK, CYP4Z1 CYP2A6 902/4885CYP2E1 12/4885CYP3A4 26/4885
US-20150250177-A1 PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS DDT, ACHE, PTMS CYP2A6 457/4885CYP2E1 111/4885CYP3A4 98/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.