SCHEMBL17420137

SCHEMBL17420137

O=C(Nc1ccc(OC(F)(F)F)cc1)N[C@H]1CC[C@H](Oc2ccc(C(=O)NO)cc2)CC1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 20/20 0.83
FAAH O00519 14/20 0.83
RAF1 P04049 1/20 0.83
AADAC P22760 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17420136 1.00 EPHX2 (0.83) EPHX2FAAHRAF1AADAC
SCHEMBL15612039 0.91 EPHX2 (1.00) EPHX2FAAHRAF1AADAC
SCHEMBL15271834 0.91 EPHX2 (1.00) EPHX2FAAHRAF1AADAC
SCHEMBL15612306 0.91 EPHX2 (1.00) EPHX2FAAHRAF1AADAC
SCHEMBL23340590 0.90 EPHX2 (0.71) EPHX2FAAHRAF1AADAC
SCHEMBL15612815 0.89 EPHX2 (1.00) EPHX2FAAHRAF1AADAC
SCHEMBL4256246 0.89 EPHX2 (1.00) EPHX2FAAHRAF1AADAC
SCHEMBL4256244 0.89 EPHX2 (1.00) EPHX2FAAHRAF1AADAC
SCHEMBL17420143 0.89 EPHX2 (0.79) EPHX2FAAHRAF1AADAC
SCHEMBL17420144 0.89 EPHX2 (0.79) EPHX2FAAHRAF1AADAC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260130877-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS THE REGENTS OF THE UNIV OF CALIFORNIA (US) 2026-05-14 US claimed
US-20230301949-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS CHIBA UNIVERSITY (JP) 2023-09-28 US claimed
US-11723929-B2 Methods of improving cell-based therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-08-15 US claimed
US-11690837-B2 Methods of improving cell-based therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-07-04 US claimed
US-11564914-B2 Methods of treating bone loss THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-01-31 US claimed
US-20220202744-A1 METHODS OF TREATING MENTAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2022-06-30 US claimed
US-20210145891-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2021-05-20 US claimed
US-20200306232-A1 METHODS OF TREATING BONE LOSS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-10-01 US claimed
US-20190125696-A1 METHODS OF TREATING MENTAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-05-02 US claimed
WO-2018231702-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-12-20 WO claimed
US-20180200244-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-19 US claimed
US-20180185309-A1 METHODS AND COMPOSITIONS FOR TREATING NEPHROPATHY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-05 US claimed
US-20260130877-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS THE REGENTS OF THE UNIV OF CALIFORNIA (US) 2026-05-14 US disclosed
US-12357598-B2 Treatment of neurodevelopmental disorders THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-07-15 US disclosed
US-20230301949-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS CHIBA UNIVERSITY (JP) 2023-09-28 US disclosed
US-11723929-B2 Methods of improving cell-based therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-08-15 US disclosed
US-20180200244-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-19 US disclosed
US-20180185309-A1 METHODS AND COMPOSITIONS FOR TREATING NEPHROPATHY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-05 US disclosed
WO-2017214394-A2 METHODS OF TREATING BONE LOSS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-12-14 WO disclosed
US-20160008342-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-01-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200306232-A1 METHODS OF TREATING BONE LOSS EPHX1, NCEH1, SOST EPHX2 4/4885FAAH 61/4885RAF1 3438/4885
US-20230301949-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS FABP7, ADH1B, ELOVL1 EPHX2 51/4885FAAH 33/4885RAF1 3702/4885
US-20160008342-A1 METHODS OF IMPROVING CELL-BASED THERAPY ELOVL1, ELOVL3, IL2 EPHX2 127/4885FAAH 223/4885RAF1 4122/4885
US-11723929-B2 Methods of improving cell-based therapy EPHX1, EPHX2, NCEH1 EPHX2 2/4885FAAH 13/4885RAF1 3766/4885
US-20180200244-A1 METHODS OF IMPROVING CELL-BASED THERAPY ELOVL1, ELOVL3, IL2 EPHX2 127/4885FAAH 223/4885RAF1 4122/4885
US-20220202744-A1 METHODS OF TREATING MENTAL DISORDERS FAAH, EPHX1, FAAH2 EPHX2 4/4885FAAH 1/4885RAF1 2980/4885
US-12357598-B2 Treatment of neurodevelopmental disorders FABP7, ADH1B, ELOVL1 EPHX2 51/4885FAAH 33/4885RAF1 3702/4885
US-20260130877-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS EED, ICOS, FABP7 EPHX2 10/4885FAAH 213/4885RAF1 4737/4885
US-11690837-B2 Methods of improving cell-based therapy ELOVL1, ELOVL3, IL2 EPHX2 127/4885FAAH 223/4885RAF1 4122/4885
US-11564914-B2 Methods of treating bone loss EPHX1, NCEH1, SOST EPHX2 4/4885FAAH 61/4885RAF1 3438/4885
US-20180185309-A1 METHODS AND COMPOSITIONS FOR TREATING NEPHROPATHY GLS, REN, SLC5A2 EPHX2 3353/4885FAAH 4685/4885RAF1 1979/4885
US-20210145891-A1 METHODS OF IMPROVING CELL-BASED THERAPY EPHX1, EPHX2, NCEH1 EPHX2 2/4885FAAH 13/4885RAF1 3766/4885
US-20190125696-A1 METHODS OF TREATING MENTAL DISORDERS FAAH, EPHX1, FAAH2 EPHX2 4/4885FAAH 1/4885RAF1 2980/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.