SCHEMBL4256244

SCHEMBL4256244

O=C(Nc1ccc(OC(F)(F)F)cc1)NC1CCC(Oc2ccc(C(=O)O)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 20/20 1.00
FAAH O00519 14/20 1.00
AADAC P22760 1/20 0.80
RAF1 P04049 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4256246 1.00 EPHX2 (1.00) EPHX2FAAHAADACRAF1
SCHEMBL15612815 1.00 EPHX2 (1.00) EPHX2FAAHAADACRAF1
SCHEMBL22223914 0.91 EPHX2 (0.84) EPHX2FAAHAADACRAF1
SCHEMBL22223736 0.91 EPHX2 (0.84) EPHX2FAAHAADACRAF1
SCHEMBL31114553 0.91 EPHX2 (0.83) EPHX2FAAHAADACRAF1
SCHEMBL19358914 0.90 EPHX2 (1.00) EPHX2FAAHAADACRAF1
SCHEMBL19358879 0.90 EPHX2 (1.00) EPHX2FAAHAADACRAF1
SCHEMBL31114447 0.90 EPHX2 (1.00) EPHX2FAAHAADACRAF1
SCHEMBL19358878 0.90 EPHX2 (1.00) EPHX2FAAHAADACRAF1
SCHEMBL17420136 0.89 EPHX2 (0.83) EPHX2FAAHAADACRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 138 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260130877-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS THE REGENTS OF THE UNIV OF CALIFORNIA (US) 2026-05-14 US claimed
US-12485107-B2 Methods for the prevention or treatment of cytokine storm BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2025-12-02 US claimed
CN-119528936-A Ballon Sha Wei derivative and application thereof 深圳安泰维生物医药有限公司 2025-02-28 CN claimed
CN-118557564-A Application of 14, 15-epoxy eicosatrienoic acid in preparation of medicine for treating traumatic brain injury 人工智能与数字经济广东省实验室(广州) 2024-08-30 CN claimed
CN-117731650-A Method for preventing and treating intestinal injury caused by high-sugar diet and application thereof 重庆医科大学 2024-03-22 CN claimed
US-20240082211-A1 SOLUBLE EPOXIDE HYDROLASE AS A TARGET FOR OCULAR DISEASES INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION 2024-03-14 US claimed
US-20230375561-A1 METHODS FOR IDENTIFICATION, STRATIFICATION, AND TREATMENT OF CNS DISEASES KADDURAH DAOUK RIMA F (US) 2023-11-23 US claimed
US-20230301949-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS CHIBA UNIVERSITY (JP) 2023-09-28 US claimed
US-11723929-B2 Methods of improving cell-based therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-08-15 US claimed
US-11690837-B2 Methods of improving cell-based therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-07-04 US claimed
CN-107132293-B Novel method for rapidly detecting EETs of brain tissues 南方医科大学 2020-12-15 CN claimed
US-20200306232-A1 METHODS OF TREATING BONE LOSS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-10-01 US claimed
US-10383835-B2 Treatment of inflammatory disorders in non-human mammals THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-08-20 US claimed
US-20190125696-A1 METHODS OF TREATING MENTAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-05-02 US claimed
WO-2018231702-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-12-20 WO claimed
US-20180200244-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-19 US claimed
US-20180185309-A1 METHODS AND COMPOSITIONS FOR TREATING NEPHROPATHY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-05 US claimed
EP-2846825-A1 TREATMENT OF INFLAMMATORY DISORDERS IN NON-HUMAN MAMMALS The Regents of The University of California (US) 2015-03-18 EP claimed
WO-2013138118-A1 TREATMENT OF INFLAMMATORY DISORDERS IN NON-HUMAN MAMMALS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-09-19 WO claimed
US-20090023731-A1 SOLUBLE EPOXIDE HYDROLASE INHIBITORS ARETE THERAPEUTICS, INC. 2009-01-22 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200306232-A1 METHODS OF TREATING BONE LOSS EPHX1, NCEH1, SOST EPHX2 4/4885FAAH 61/4885AADAC 3264/4885
US-20240082211-A1 SOLUBLE EPOXIDE HYDROLASE AS A TARGET FOR OCULAR DISEASES EPHX1, ALDH1A2, EPHX2 EPHX2 3/4885FAAH 30/4885AADAC 1919/4885
US-20230301949-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS FABP7, ADH1B, ELOVL1 EPHX2 51/4885FAAH 33/4885AADAC 717/4885
US-20090023731-A1 SOLUBLE EPOXIDE HYDROLASE INHIBITORS EPHX1, EPHX2, NCEH1 EPHX2 2/4885FAAH 12/4885AADAC 2120/4885
US-11723929-B2 Methods of improving cell-based therapy EPHX1, EPHX2, NCEH1 EPHX2 2/4885FAAH 13/4885AADAC 1463/4885
US-20180200244-A1 METHODS OF IMPROVING CELL-BASED THERAPY ELOVL1, ELOVL3, IL2 EPHX2 127/4885FAAH 223/4885AADAC 873/4885
US-20260130877-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS EED, ICOS, FABP7 EPHX2 10/4885FAAH 213/4885AADAC 2390/4885
US-11690837-B2 Methods of improving cell-based therapy ELOVL1, ELOVL3, IL2 EPHX2 127/4885FAAH 223/4885AADAC 873/4885
US-12485107-B2 Methods for the prevention or treatment of cytokine storm TNF, PTGES2, IL2 EPHX2 13/4885FAAH 16/4885AADAC 1640/4885
US-20180185309-A1 METHODS AND COMPOSITIONS FOR TREATING NEPHROPATHY GLS, REN, SLC5A2 EPHX2 3353/4885FAAH 4685/4885AADAC 4383/4885
US-20190125696-A1 METHODS OF TREATING MENTAL DISORDERS FAAH, EPHX1, FAAH2 EPHX2 4/4885FAAH 1/4885AADAC 871/4885
US-20230375561-A1 METHODS FOR IDENTIFICATION, STRATIFICATION, AND TREATMENT OF CNS DISEASES SLC25A20, CPT2, NDUFAB1 EPHX2 1139/4885FAAH 69/4885AADAC 747/4885
US-10383835-B2 Treatment of inflammatory disorders in non-human mammals EPHX1, SERPINB1, PTGES EPHX2 13/4885FAAH 11/4885AADAC 539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.