SCHEMBL17524928

SCHEMBL17524928

O=C1Nc2ncccc2C12CCN(c1ccc(I)c(Oc3ccccc3)c1)CC2

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.37
CALCA P06881 8/20 0.36
EGLN1 Q9GZT9 1/20 0.35
HTR1A P08908 5/20 0.35
HTR2A P28223 5/20 0.35
HTR7 P34969 5/20 0.35
SCN9A Q15858 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CALCRL Q16602 2/20 0.33
RIPK1 Q13546 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524873 0.89 HTR6 (0.38) HTR6CALCAEGLN1HTR1AHTR2A
SCHEMBL17524879 0.81 HTR6 (0.34) HTR6CALCAEGLN1
SCHEMBL17525019 0.79 MAPK1 (0.41) HTR6CALCAHTR1AHTR2AHTR7
SCHEMBL17524951 0.78 LTA4H (0.38) HTR6CALCAHTR1AHTR2AHTR7
SCHEMBL17524907 0.78 MALT1 (0.41) CALCAEGLN1CALCRL
SCHEMBL17524933 0.78 CALCA (0.40) HTR6CALCAEGLN1HTR1AHTR2A
SCHEMBL17524881 0.78 CRHR1 (0.33) HTR6CALCAEGLN1CALCRLRIPK1
SCHEMBL17525080 0.77 LRRK2 (0.39) HTR6CALCAEGLN1HTR1AHTR2A
SCHEMBL17524901 0.77 ADRA2B (0.40) HTR6CALCAEGLN1HTR1AHTR2A
SCHEMBL17524942 0.77 ADRA2B (0.40) HTR6CALCAEGLN1HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed