SCHEMBL17524951

SCHEMBL17524951

Nc1ccc(N2CCC3(CC2)C(=O)Nc2ncccc23)cc1OCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.38
MAPK14 Q16539 1/20 0.38
CALCA P06881 7/20 0.38
LRRK2 Q5S007 5/20 0.37
GRM5 P41594 1/20 0.36
GRM3 Q14832 1/20 0.36
HTR6 P50406 3/20 0.36
HTR1A P08908 2/20 0.36
HTR2A P28223 2/20 0.36
HTR7 P34969 2/20 0.36
TNKS2 Q9H2K2 1/20 0.36
CALCRL Q16602 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17525080 0.90 LRRK2 (0.39) CALCALRRK2HTR6HTR1AHTR2A
SCHEMBL17524942 0.87 ADRA2B (0.40) CALCAHTR6HTR1AHTR2AHTR7
SCHEMBL17524873 0.87 HTR6 (0.38) CALCAHTR6HTR1AHTR2AHTR7
SCHEMBL17524933 0.85 CALCA (0.40) CALCAHTR6HTR1AHTR2AHTR7
SCHEMBL17524957 0.85 CALCA (0.38) CALCAHTR6HTR1AHTR2AHTR7
SCHEMBL17524946 0.85 CALCRL (0.38) CALCAHTR6HTR1AHTR2AHTR7
SCHEMBL17524938 0.80 HTR7 (0.45) CALCAHTR6HTR1AHTR2AHTR7
SCHEMBL17524935 0.80 GAA (0.44) CALCAHTR6HTR1AHTR2AHTR7
SCHEMBL17524940 0.80 CALCA (0.40) CALCAHTR6HTR1AHTR2AHTR7
SCHEMBL17524928 0.78 HTR6 (0.37) CALCAHTR6HTR1AHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed