SCHEMBL17524946

SCHEMBL17524946

Nc1ccc(N2CCC3(CC2)C(=O)Nc2ncccc23)cc1OCC(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 6/20 0.38
CALCA P06881 4/20 0.38
ADRA2B P18089 1/20 0.36
PTPN11 Q06124 1/20 0.36
IDH1 O75874 3/20 0.35
HTR1A P08908 2/20 0.34
HTR2A P28223 2/20 0.34
HTR7 P34969 2/20 0.34
HTR6 P50406 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
G6PD P11413 1/20 0.34
ALOX15 P16050 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524909 0.90 ADRA1A (0.38) CALCRLCALCAADRA2BIDH1ADRA1D
SCHEMBL17524942 0.87 ADRA2B (0.40) CALCRLCALCAADRA2BIDH1HTR1A
SCHEMBL17524933 0.85 CALCA (0.40) CALCRLCALCAIDH1HTR1AHTR2A
SCHEMBL17524951 0.85 LTA4H (0.38) CALCRLCALCAHTR1AHTR2AHTR7
SCHEMBL17524957 0.85 CALCA (0.38) CALCRLCALCAIDH1HTR1AHTR2A
SCHEMBL17524873 0.83 HTR6 (0.38) CALCRLCALCAHTR1AHTR2AHTR7
SCHEMBL17524940 0.82 CALCA (0.40) CALCRLCALCAPTPN11HTR1AHTR2A
SCHEMBL17524935 0.80 GAA (0.44) CALCRLCALCAHTR1AHTR2AHTR7
SCHEMBL17524938 0.80 HTR7 (0.45) CALCRLCALCAHTR1AHTR2AHTR7
SCHEMBL17524901 0.78 ADRA2B (0.40) CALCRLCALCAADRA2BHTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed