SCHEMBL17599342

SCHEMBL17599342

O=C(O)c1cccc(-c2ccc(NS(=O)(=O)c3cc(F)cc(F)c3F)c3ccccc23)c1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 5/20 0.45
FABP5 Q01469 3/20 0.45
KMT2A Q03164 1/20 0.45
ACLY P53396 10/20 0.45
PTK2B Q14289 2/20 0.43
SLC16A3 O15427 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17599319 0.84 ACLY (0.46) FABP4FABP5KMT2AACLYPTK2B
SCHEMBL17599400 0.84 KMT2A (0.49) FABP4FABP5KMT2AACLYPTK2B
SCHEMBL17599337 0.82 PTK2B (0.50) FABP4FABP5KMT2AACLYPTK2B
SCHEMBL17599310 0.82 PTK2B (0.53) FABP4FABP5KMT2AACLYPTK2B
SCHEMBL17599402 0.82 BRD4 (0.52) FABP4FABP5KMT2AACLYPTK2B
SCHEMBL17599317 0.80 FABP4 (0.52) FABP4FABP5KMT2AACLYPTK2B
SCHEMBL17599379 0.79 ACLY (0.54) FABP4KMT2AACLYPTK2BSLC16A3
SCHEMBL17599360 0.78 ITGA1 (0.56) FABP4FABP5KMT2AACLYPTK2B
SCHEMBL17599340 0.78 SLC16A3 (0.58) FABP4KMT2AACLYPTK2BSLC16A3
SCHEMBL17599403 0.77 WDR5 (0.49) FABP4KMT2AACLYPTK2BSLC16A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2998294-A1 Naphthyl sulfonamide phenyl derivatives as KEAP-1 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders SANOFI (FR) 2016-03-23 EP disclosed
EP-2998294-A1 Naphthyl sulfonamide phenyl derivatives as KEAP-1 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders SANOFI (FR) 2016-03-23 EP disclosed