SCHEMBL1764951

SCHEMBL1764951

COc1ccccc1C(=O)/C=C/c1cccc(OC)c1OC

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.70
ABCG2 Q9UNQ0 1/20 0.66
MAOB P27338 4/20 0.65
ALOX5 P09917 2/20 0.65
CYP1A1 P04798 1/20 0.65
CYP1A2 P05177 1/20 0.65
CYP2D6 P10635 1/20 0.65
AR P10275 2/20 0.64
NR1H4 Q96RI1 1/20 0.63
TRPM8 Q7Z2W7 1/20 0.61
ALDH1A1 P00352 2/20 0.58
LMNA P02545 2/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
KDM4E B2RXH2 1/20 0.58
MEN1 O00255 1/20 0.58
POLB P06746 1/20 0.58
GAA P10253 1/20 0.58
MAPT P10636 1/20 0.58
PKM P14618 1/20 0.58
HPGD P15428 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4864045 0.93 NFE2L2 (0.72) NFE2L2ABCG2MAOBALOX5CYP1A1
SCHEMBL5084423 0.90 MAOB (0.80) NFE2L2ABCG2MAOBALOX5CYP1A1
SCHEMBL5084427 0.90 MAOB (0.80) NFE2L2ABCG2MAOBALOX5CYP1A1
SCHEMBL7096835 0.89 NFE2L2 (0.63) NFE2L2MAOBALOX5CYP1A1CYP1A2
SCHEMBL11073098 0.88 NFE2L2 (0.59) NFE2L2ABCG2MAOBALOX5CYP1A1
SCHEMBL4535102 0.88 AR (0.80) NFE2L2ABCG2MAOBCYP1A1CYP1A2
SCHEMBL7097185 0.87 ALDH1A1 (0.68) NFE2L2MAOBALOX5CYP1A1CYP1A2
SCHEMBL7099531 0.87 PTPN1 (0.61) NFE2L2MAOBALOX5CYP1A1CYP1A2
SCHEMBL27794060 0.87 NFE2L2 (0.60) NFE2L2ABCG2MAOBALOX5CYP1A1
SCHEMBL4026900 0.85 LMNA (0.78) NFE2L2ABCG2MAOBALOX5CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115624544-B Application of chalcone analogue as active substance in preparation of antitumor drugs 甘肃中医药大学 2025-01-24 CN claimed
EP-0021000-B1 SUBSTITUTED ACETOPHENONES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-02-22 EP claimed
EP-4598515-A1 PHYTOCHEMICAL FORMULATIONS FOR TREATING STRESS AND ANXIETY GBS Global Biopharma, Inc. (CA) 2025-08-13 EP disclosed
EP-4429763-A1 COMPOSITIONS AND METHODS FOR TREATING BLEEDING AND BLEEDING DISORDERS Yewsavin, Inc. (US) 2024-09-18 EP disclosed
EP-2984072-B1 SYNTHETIC ANALOGUES OF XANTHOHUMOL UNIV PISA (IT) 2024-05-29 EP disclosed
WO-2024054462-A1 PHYTOCHEMICAL FORMULATIONS FOR TREATING STRESS AND ANXIETY GBS GLOBAL BIOPHARMA, INC. (CA) 2024-03-14 WO disclosed
WO-2023086388-A1 COMPOSITIONS AND METHODS FOR TREATING BLEEDING AND BLEEDING DISORDERS YewSavin, Inc. (US) 2023-05-19 WO disclosed
CN-115624544-A Application of chalcone analogue as active substance in preparation of antitumor drugs 甘肃中医药大学 2023-01-20 CN disclosed
US-9617213-B2 Synthetic analogues of xanthohumol UNIVERSITA' DI PISA (IT) 2017-04-11 US disclosed
US-20160075652-A1 SYNTHETIC ANALOGUES OF XANTHOHUMOL AZIENDA OSPEDALIERA DI REGGIO EMILIA ARCISPEDALE S. MARIA NUOVA IRCCS (IT) 2016-03-17 US disclosed
US-20110124721-A1 METHODS OF TREATING TRAUMATIC BRAIN INJURY BY ADMINISTERING BAICALEIN PREPARATION NATIONAL DEFENSE MEDICAL CENTER (TW) 2011-05-26 US disclosed
US-20100222421-A1 Usage of Baicalein in the Preparation of a Pharmaceutical Composition for the Treatment of Traumatic Brain Injury NATIONAL DEFENSE MEDICAL CENTER (TW) 2010-09-02 US disclosed
US-20080287374-A1 BREAST CANCER-RESISTANT PROTEIN INHIBITOR KABUSHIKI KAISHA YAKULT HONSHA (JP) 2008-11-20 US disclosed
EP-1888174-A1 USE OF CHALCONES FOR THE TREATMENT OF VIRAL DISORDERS Johnson and Johnson Consumer Companies, Inc. (US) 2008-02-20 EP disclosed
US-7326734-B2 Treatment of bladder and urinary tract cancers THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2008-02-05 US disclosed
WO-2006127539-A1 USE OF CHALCONES FOR THE TREATMENT OF VIRAL DISORDERS JOHNSON & JOHNSON CONSUMER COMPANIES, INC. (US) 2006-11-30 WO disclosed
US-20060135445-A1 Breast cancer-resistant protein inhibitor KABUSHIKI KAISHA YAKULT HONSHA (JP) 2006-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160075652-A1 SYNTHETIC ANALOGUES OF XANTHOHUMOL XDH, XPA, NR1H3 NFE2L2 3341/4885ABCG2 1193/4885MAOB 1648/4885
US-20060135445-A1 Breast cancer-resistant protein inhibitor ABCC1, BCR, BRCA1 NFE2L2 1167/4885ABCG2 8/4885MAOB 3350/4885
US-20080287374-A1 BREAST CANCER-RESISTANT PROTEIN INHIBITOR ABCC1, BCR, BRCA1 NFE2L2 1167/4885ABCG2 8/4885MAOB 3350/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.