SCHEMBL18179853

SCHEMBL18179853

COc1cc(CC[PH](c2ccccc2)(c2ccccc2)c2ccccc2)cc(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.46
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
CALM1 P0DP23 3/20 0.44
AKR1B1 P15121 1/20 0.44
ABCB1 P08183 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
TACR1 P25103 2/20 0.42
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
MAOB P27338 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
GAA P10253 1/20 0.40
LTA4H P09960 1/20 0.39
CA4 P22748 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28031835 0.84 LTA4H (0.53) ABCB1L3MBTL1SIGMAR1LTA4HCA4
SCHEMBL5083307 0.82 TSHR (0.47) CYP19A1TSHRMAPK1CALM1AKR1B1
Bromide SCHEMBL16180511 0.81 TSHR (0.46) CYP19A1TSHRMAPK1CALM1AKR1B1
SCHEMBL18179854 0.80 MEN1 (0.49) L3MBTL1MAOBGAALTA4H
SCHEMBL1972535 0.77 CYP19A1 (0.66) CYP19A1TSHRMAPK1CALM1AKR1B1
SCHEMBL13086387 0.75 ALDH1A1 (0.46) TSHRMAOBSIGMAR1
Hydrochloric Acid SCHEMBL28127090 0.73 ALDH1A1 (0.44) L3MBTL1MAOBGAA
SCHEMBL5973660 0.72 MAOB (0.57) CALM1ABCB1MAOBSIGMAR1
Bromide SCHEMBL28593166 0.72 TACR1 (0.48) TSHRMAPK1ABCB1TACR1MAOB
SCHEMBL9491787 0.72 CYP19A1 (0.68) CYP19A1TSHRCALM1AKR1B1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10004722-B2 Method for treating hepatic encephalopathy or a disease associated with free radical mediate stress and oxidative stress with novel functionalized 1,3-benzene diols KANNALIFE SCIENCES, INC. (US) 2018-06-26 US disclosed
US-20170157097-A1 METHOD FOR TREATING HEPATIC ENCEPHALOPATHY OR A DISEASE ASSOCIATED WITH FREE RADICAL MEDIATE STRESS AND OXIDATIVE STRESS WITH NOVEL FUNCTIONALIZED 1,3-BENZENE DIOLS KANNALIFE SCIENCES, INC. 2017-06-08 US disclosed
US-20170157097-A1 METHOD FOR TREATING HEPATIC ENCEPHALOPATHY OR A DISEASE ASSOCIATED WITH FREE RADICAL MEDIATE STRESS AND OXIDATIVE STRESS WITH NOVEL FUNCTIONALIZED 1,3-BENZENE DIOLS KANNALIFE SCIENCES, INC. 2017-06-08 US disclosed
US-9611213-B2 Functionalized 1,3-benzene diols and their method of use for the treatment of hepatic encephalopathy KANNALIFE SCIENCES, INC. (US) 2017-04-04 US disclosed
US-20160311769-A1 NOVEL FUNCTIONALIZED 1,3-BENZENE DIOLS AND THEIR METHOD OF USE FOR THE TREATMENT OF HEPATIC ENCEPHALOPTHY KANNALIFE SCIENCES, INC. 2016-10-27 US disclosed
US-20150202335-A1 TARGETED MOLECULAR IMAGING PROBE AND METHOD FOR IN VIVO MOLECULAR IMAGING SHEN BAOZHONG (CN) 2015-07-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170157097-A1 METHOD FOR TREATING HEPATIC ENCEPHALOPATHY OR A DISEASE ASSOCIATED WITH FREE RADICAL MEDIATE STRESS AND OXIDATIVE STRESS WITH NOVEL FUNCTIONALIZED 1,3-BENZENE DIOLS TXNRD2, KEAP1, GOT2 CYP19A1 1518/4885TSHR 3175/4885MAPK1 1444/4885
US-20160311769-A1 NOVEL FUNCTIONALIZED 1,3-BENZENE DIOLS AND THEIR METHOD OF USE FOR THE TREATMENT OF HEPATIC ENCEPHALOPTHY EPHX1, DBH, EPHX2 CYP19A1 2594/4885TSHR 3038/4885MAPK1 3104/4885
US-20150202335-A1 TARGETED MOLECULAR IMAGING PROBE AND METHOD FOR IN VIVO MOLECULAR IMAGING GJB2, GJA1, GAP43 CYP19A1 4722/4885TSHR 4266/4885MAPK1 1114/4885
US-10004722-B2 Method for treating hepatic encephalopathy or a disease associated with free radical mediate stress and oxidative stress with novel functionalized 1,3-benzene diols TXNRD2, KEAP1, GOT2 CYP19A1 1518/4885TSHR 3175/4885MAPK1 1444/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.