SCHEMBL196828

SCHEMBL196828

CN(C)/C(N)=N/CCC[C@H](N)C(=O)O

nearest known ligand 0.79

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 10/20 0.79
NOS1 P29475 9/20 0.67
NOS3 P29474 5/20 0.67
CYP2C19 P33261 3/20 0.67
MEN1 O00255 1/20 0.67
KMT2A Q03164 1/20 0.67
CYP1A2 P05177 2/20 0.66
TSHR P16473 2/20 0.66
GLA P06280 1/20 0.66
NFKB1 P19838 1/20 0.66
APEX1 P27695 1/20 0.66
DDAH1 O94760 6/20 0.63
THPO P40225 1/20 0.61
CYP3A4 P08684 1/20 0.60
BLM P54132 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13484050 1.00 NOS2 (0.79) NOS2NOS1NOS3CYP2C19MEN1
SCHEMBL995818 1.00 NOS2 (0.79) NOS2NOS1NOS3CYP2C19MEN1
SCHEMBL14843061 1.00 NOS2 (0.79) NOS2NOS1NOS3CYP2C19MEN1
SCHEMBL31436337 0.89 NOS2 (0.68) NOS2NOS1NOS3CYP2C19MEN1
Hydrochloric Acid SCHEMBL30114268 0.87 NOS2 (0.66) NOS2NOS1NOS3CYP2C19MEN1
L-Nio SCHEMBL15944942 0.80 NOS2 (1.00) NOS2NOS1NOS3CYP2C19MEN1
Arginine SCHEMBL43261 0.80 NOS2 (1.00) NOS2NOS1NOS3CYP2C19MEN1
Arginine SCHEMBL30577923 0.80 NOS2 (1.00) NOS2NOS1NOS3CYP2C19MEN1
Arginine SCHEMBL288835 0.80 NOS2 (1.00) NOS2NOS1NOS3CYP2C19MEN1
Arginine SCHEMBL288993 0.80 NOS2 (1.00) NOS2NOS1NOS3CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 109 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250011774-A1 ANTISENSE COMPOUNDS AND METHODS FOR TARGETING CUG REPEATS ENTRADA THERAPEUTICS, INC. 2025-01-09 US claimed
EP-4359006-A1 ANTISENSE COMPOUNDS AND METHODS FOR TARGETING CUG REPEATS Entrada Therapeutics, Inc. (US) 2024-05-01 EP claimed
WO-2023185709-A1 MARKER COMBINATION FOR DIAGNOSING ADVANCED COLORECTAL TUMOR, AND APPLICATION THEREOF 武汉迈特维尔医学科技有限公司 2023-10-05 WO claimed
WO-2023192510-A1 β-CATENIN ANTIBODIES ENTRADA THERAPEUTICS, INC. (US) 2023-10-05 WO claimed
US-20230027739-A1 ANTIGEN-BINDING AND ANTIGEN DEGRADATION CONSTRUCTS ENTRADA THERAPEUTICS, INC. 2023-01-26 US claimed
WO-2022271818-A1 ANTISENSE COMPOUNDS AND METHODS FOR TARGETING CUG REPEATS ENTRADA THERAPEUTICS, INC. (US) 2022-12-29 WO claimed
CN-106370753-A Identification and analysis method for coronary heart disease urine metabolic markers 王喜军 2017-02-01 CN claimed
US-20260098262-A9 COMPOUNDS AND METHODS FOR SKIPPING EXON 44 IN DUCHENNE MUSCULAR DYSTROPHY ENTRADA THERAPEUTICS INC (US) 2026-04-09 US disclosed
US-20260028630-A1 HYBRID OLIGONUCLEOTIDES ENTRADA THERAPEUTICS INC (US) 2026-01-29 US disclosed
US-20250289851-A1 CYCLIC PEPTIDES FOR DELIVERING THERAPEUTICS ENTRADA THERAPEUTICS, INC. 2025-09-18 US disclosed
US-20250243244-A1 CYCLIC CELL PENETRATING PEPTIDES ENTRADA THERAPEUTICS, INC. 2025-07-31 US disclosed
US-20250228953-A1 INTRACELLULAR TARGETING OF OLIGONUCLEOTIDES ENTRADA THERAPEUTICS, INC. 2025-07-17 US disclosed
WO-2025125621-A1 CANCER-ASSOCIATED PROTEIN-TARGETED STRONG OR COVALENTLY BINDING PRECURSOR COMPOUNDS AND RADIOTRACERS RADIOVAXX GMBH (DE) 2025-06-19 WO disclosed
US-20070149446-A1 Tamandarin analogs and fragments thereof and methods of making and using THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA CENTER FOR TECHNOLOGY TRANSFER (US) 2007-06-28 US disclosed
US-20060035854-A1 Compositions and methods for coating medical devices GOLDSTEIN STEVEN 2006-02-16 US disclosed
EP-0910301-A4 COMPOSITIONS AND METHODS FOR COATING MEDICAL DEVICES UNIV MICHIGAN (US) 2004-10-27 EP disclosed
US-6358699-B1 REMOVING INTERFERING COMPONENTS FROM SAMPLE, CONTACTING WITH DIMETHYLARGININE DIMETHYLAMINO-HYDROLASE TO HYDROLYZE DIMETHYLARGININE TO CITRULLINE, SPECTROPHOTOMETRICALLY DETERMINING CITRULLINE COOKE PHARMA 2002-03-19 US disclosed
US-6143037-A MEDICAL EQUIPMENT COATED WITH A BIOCOMPATIBLE AND BIODEGRADABLE POLMERIC MATRIX AND A NULEIC ACID THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2000-11-07 US disclosed
EP-0910301-A1 COMPOSITIONS AND METHODS FOR COATING MEDICAL DEVICES THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 1999-04-28 EP disclosed
WO-1997047254-A1 COMPOSITIONS AND METHODS FOR COATING MEDICAL DEVICES THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 1997-12-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260028630-A1 HYBRID OLIGONUCLEOTIDES RNGTT, BCDIN3D, RNMT NOS2 4732/4885NOS1 4621/4885NOS3 3842/4885
US-20250228953-A1 INTRACELLULAR TARGETING OF OLIGONUCLEOTIDES MAN1B1, RNASE1, ERAP1 NOS2 4785/4885NOS1 4764/4885NOS3 4756/4885
US-20250243244-A1 CYCLIC CELL PENETRATING PEPTIDES SLC47A1, SLC47A2, VIP NOS2 2084/4885NOS1 2445/4885NOS3 2929/4885
US-20260098262-A9 COMPOUNDS AND METHODS FOR SKIPPING EXON 44 IN DUCHENNE MUSCULAR DYSTROPHY UTRN, SMN1; SMN2, UPF1 NOS2 4699/4885NOS1 4569/4885NOS3 4351/4885
US-20230027739-A1 ANTIGEN-BINDING AND ANTIGEN DEGRADATION CONSTRUCTS PRCP, TAP1, DNPEP NOS2 4518/4885NOS1 4467/4885NOS3 4611/4885
US-20250011774-A1 ANTISENSE COMPOUNDS AND METHODS FOR TARGETING CUG REPEATS CDR2, SMN1; SMN2, ATXN2 NOS2 4568/4885NOS1 4745/4885NOS3 4787/4885
US-20250289851-A1 CYCLIC PEPTIDES FOR DELIVERING THERAPEUTICS IAPP, LNPEP, CFTR NOS2 3390/4885NOS1 3719/4885NOS3 3474/4885
US-20070149446-A1 Tamandarin analogs and fragments thereof and methods of making and using FOXM1, F3, RB1 NOS2 874/4885NOS1 595/4885NOS3 376/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.