SCHEMBL1970565

SCHEMBL1970565

FC1(F)Oc2ccc(N=C=S)cc2O1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY6 Q15077 2/20 0.37
MIF P14174 1/20 0.36
NAAA Q02083 1/20 0.36
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36
PNMT P11086 1/20 0.35
NOTUM Q6P988 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CG P48736 1/20 0.35
KIF11 P52732 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KDM4E B2RXH2 2/20 0.34
USP2 O75604 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LTA P01374 2/20 0.34
CYP3A4 P08684 2/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 2/20 0.34
P2RX3 P56373 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30298625 1.00 P2RY6 (0.37) P2RY6MIFNAAACTNNB1WNT3A
SCHEMBL10850783 0.89 P2RY6 (0.37) P2RY6MIFPNMTKIF11KDM4E
SCHEMBL11114110 0.82 P2RY6 (0.33) P2RY6MIFPNMTKDM4EUSP2
SCHEMBL11003249 0.82 MAPK1 (0.43) CTNNB1WNT3ANOTUMPIK3CAPIK3CG
SCHEMBL11000954 0.79 PNMT (0.34) P2RY6MIFPNMTKDM4EUSP2
SCHEMBL11000092 0.78 P2RY6 (0.32) P2RY6MIFPNMTKDM4EUSP2
SCHEMBL9428400 0.77 P2RY6 (0.37) P2RY6MIFPNMTKDM4EUSP2
SCHEMBL10451237 0.71 MAPK1 (0.43) KIF11CYP3A4TDP1
SCHEMBL276124 0.70 ADRA2A (0.53) P2RY6MIFPNMTNPC1RAB9A
SCHEMBL1019410 0.70 HTR3E (0.53) P2RY6MIFPNMTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259267-B2 Difluorobenzo-1,3-dioxoles LANXESS DEUTSCHLAND GMBH (DE) 2007-08-21 US claimed
US-20050272811-A1 Difluorobenzo-1,3-dioxoles LANXESS DEUTSCHLAND GMBH (DE) 2005-12-08 US claimed
EP-1595875-A2 Isothiocyanato-2,2-difluoro-1,3-benzodioxoles Lanxess Deutschland GmbH (DE) 2005-11-16 EP claimed
EP-4139286-B1 SUBSTITUTED AMINOTHIAZOLES AS DGKZETA INHIBITORS FOR IMMUNE ACTIVATION BAYER AG (DE) 2025-02-26 EP disclosed
US-12018021-B2 Thiophene derivatives for the treatment of disorders caused by IgE UCB Biopharma SRL (BE) 2024-06-25 US disclosed
US-11964953-B2 Substituted aminothiazoles as DGKzeta inhibitors for immune activation BAYER AKTIENGESELLSCHAFT (DE) 2024-04-23 US disclosed
WO-2023158862-A2 STIMULATOR OF INTERFERON GENES (STING) MODULATORS, AND COMPOSITIONS AND METHODS THEREOF GEODE THERAPEUTICS INC. (US) 2023-08-24 WO disclosed
US-20230167078-A1 SUBSTITUTED AMINOTHIAZOLES AS DGKZETA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2023-06-01 US disclosed
US-20230139936-A1 SUBSTITUTED AMINOTHIAZOLES AS DGKZETA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2023-05-04 US disclosed
CN-112566910-A Thiophene derivatives for the treatment of IgE induced diseases UCB生物制药有限责任公司 2021-03-26 CN disclosed
EP-1595875-B1 Process for the preparation of isothiocyanato-2,2-difluoro-1,3-benzodioxoles SALTIGO GMBH (DE) 2011-06-22 EP disclosed
CN-100569766-C The difluoro phendioxin, the 3-dioxole LANXESS DEUTSCHLAND GMBH (DE) 2009-12-16 CN disclosed
US-7259267-B2 Difluorobenzo-1,3-dioxoles LANXESS DEUTSCHLAND GMBH (DE) 2007-08-21 US disclosed
US-20050272811-A1 Difluorobenzo-1,3-dioxoles LANXESS DEUTSCHLAND GMBH (DE) 2005-12-08 US disclosed
EP-1595875-A2 Isothiocyanato-2,2-difluoro-1,3-benzodioxoles Lanxess Deutschland GmbH (DE) 2005-11-16 EP disclosed
CN-1696126-A Process for the preparation of 5-bromo-2,2-difluorobenzo-(1,3)-dioxoles LANXESS DEUTSCHLAND GMBH (DE) 2005-11-16 CN disclosed
US-4536587-A APPLYING DIRECTLY TO HABITAT BAYER AKTIENGESELLSCHAFT (DE) 1985-08-20 US disclosed
EP-0042533-B1 SUBSTITUTED BENZOYL(THIO) UREAS, PROCESSES FOR THEIR PRODUCTION AND THEIR USE AS PESTICIDES BAYER AG (DE) 1984-03-14 EP disclosed
EP-0042533-A1 Substituted benzoyl(thio) ureas, processes for their production and their use as pesticides BAYER AG (DE) 1981-12-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230139936-A1 SUBSTITUTED AMINOTHIAZOLES AS DGKZETA INHIBITORS FOR IMMUNE ACTIVATION DGKZ, DGKA, DGKG P2RY6 1187/4885MIF 3660/4885NAAA 1783/4885
US-20230167078-A1 SUBSTITUTED AMINOTHIAZOLES AS DGKZETA INHIBITORS FOR IMMUNE ACTIVATION DGKZ, DGKA, DGKG P2RY6 1187/4885MIF 3660/4885NAAA 1783/4885
US-11964953-B2 Substituted aminothiazoles as DGKzeta inhibitors for immune activation DGKZ, DGKA, DGKG P2RY6 1187/4885MIF 3660/4885NAAA 1783/4885
US-20050272811-A1 Difluorobenzo-1,3-dioxoles BROX, DDT, CAT P2RY6 2945/4885MIF 1924/4885NAAA 2940/4885
US-12018021-B2 Thiophene derivatives for the treatment of disorders caused by IgE TSLP, CYSLTR1, CYSLTR2 P2RY6 887/4885MIF 1146/4885NAAA 3429/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.