SCHEMBL19986708

SCHEMBL19986708

Cc1cc(F)cc(NC(=O)NCCCNc2c(C)cncc2C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
SLC6A3 Q01959 1/20 0.39
NAMPT P43490 1/20 0.38
KMT2A Q03164 2/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
MEN1 O00255 1/20 0.37
MARS1 P56192 1/20 0.37
BRD4 O60885 2/20 0.37
CDK2 P24941 1/20 0.37
FLT4 P35916 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
EPHX2 P34913 1/20 0.36
LCK P06239 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986718 0.85 ALDH1A1 (0.42) KDM4ESLC6A3KMT2AMEN1CDK2
SCHEMBL19986692 0.83 NAMPT (0.38) KDM4ENAMPTKMT2ASCN10AMEN1
SCHEMBL19986619 0.82 NAMPT (0.37) KDM4ENAMPTKMT2ASCN10AHDAC3
SCHEMBL19986507 0.78 KMT2A (0.38) KDM4ESLC6A3NAMPTKMT2AMEN1
SCHEMBL19986699 0.78 LMNA (0.53) NAMPTKMT2AMEN1MARS1BRD4
SCHEMBL19986705 0.77 MARS1 (0.47) SLC6A3KMT2AMEN1MARS1ALDH1A1
SCHEMBL19986671 0.75 EPHX2 (0.49) KDM4ESLC6A3KMT2AMEN1ALDH1A1
SCHEMBL19986715 0.75 KMT2A (0.41) KDM4ENAMPTKMT2AMEN1MAPT
SCHEMBL19986631 0.75 KMT2A (0.53) NAMPTKMT2AMEN1ALDH1A1MAPT
SCHEMBL19986446 0.74 KMT2A (0.49) KDM4ESLC6A3NAMPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed