SCHEMBL20118220

SCHEMBL20118220

CCC1=NN(c2ccc(F)cc2Cl)C(=O)[C@]12CC[C@H](NC(=O)c1cnn3c(C)cc(C)nc13)CC2

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
KDM4E B2RXH2 6/20 0.50
POLB P06746 2/20 0.50
GBA1 P04062 2/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 6/20 0.42
CYP1A1 P04798 1/20 0.42
HSD17B10 Q99714 2/20 0.41
USP2 O75604 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CRHR1 P34998 2/20 0.40
CRHR2 Q13324 1/20 0.40
HSD11B1 P28845 2/20 0.40
TYK2 P29597 2/20 0.39
PDE4D Q08499 1/20 0.38
PLEC Q15149 1/20 0.38
PDE4B Q07343 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118235 0.91 ALDH1A1 (0.53) ALDH1A1KDM4EPOLBGBA1MAPT
SCHEMBL20118188 0.83 KDM4E (0.47) KDM4EHSD17B10
SCHEMBL18208702 0.82 ALDH1A1 (0.54) ALDH1A1KDM4EPOLBGBA1MAPT
SCHEMBL18208588 0.82 ALDH1A1 (0.54) ALDH1A1KDM4EPOLBGBA1MAPT
SCHEMBL18208590 0.82 ALDH1A1 (0.54) ALDH1A1KDM4EPOLBGBA1MAPT
SCHEMBL20118187 0.79 PDE4B (0.41) HPGDCRHR1CRHR2HSD11B1PDE4D
SCHEMBL20118174 0.78 CRHR1 (0.40) HPGDCRHR1CRHR2PDE4B
SCHEMBL20118407 0.78 PDE4B (0.40) CRHR1CRHR2PDE4B
SCHEMBL20118213 0.77 LMNA (0.42) HPGDCRHR1CRHR2PDE4B
SCHEMBL20118184 0.77 CRHR1 (0.39) HPGDCRHR1CRHR2PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed