SCHEMBL20118407

SCHEMBL20118407

CCC1=NN(c2ccc(F)cc2Cl)C(=O)[C@]12CC[C@H](NC(=O)c1cnc3ccccc3n1)CC2

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 6/20 0.40
CRHR1 P34998 2/20 0.39
CRHR2 Q13324 1/20 0.39
HTR1A P08908 2/20 0.37
NTRK1 P04629 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118174 0.84 CRHR1 (0.40) PDE4BCRHR1CRHR2
SCHEMBL20118213 0.83 LMNA (0.42) PDE4BCRHR1CRHR2HTR1A
SCHEMBL20118187 0.81 PDE4B (0.41) PDE4BCRHR1CRHR2
SCHEMBL20118184 0.81 CRHR1 (0.39) PDE4BCRHR1CRHR2
SCHEMBL20118188 0.79 KDM4E (0.47)
SCHEMBL20118220 0.78 ALDH1A1 (0.50) PDE4BCRHR1CRHR2
SCHEMBL20118169 0.77 P2RX7 (0.35) CRHR1CRHR2
SCHEMBL20118172 0.77 P2RX7 (0.35) CRHR1CRHR2
SCHEMBL20118191 0.76 CRHR1 (0.43) PDE4BCRHR1CRHR2
SCHEMBL20118231 0.74 CRHR1 (0.37) CRHR1CRHR2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed