SCHEMBL20118213

SCHEMBL20118213

CCC1=NN(c2ccc(F)cc2Cl)C(=O)[C@]12CC[C@H](NC(=O)c1cccc3nccnc13)CC2

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
ESR1 P03372 1/20 0.42
TNKS2 Q9H2K2 8/20 0.41
CRHR1 P34998 3/20 0.40
CRHR2 Q13324 1/20 0.40
TNKS O95271 4/20 0.40
PDE4B Q07343 6/20 0.39
HPGD P15428 1/20 0.38
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
HTR7 P34969 1/20 0.36
HTR6 P50406 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118187 0.91 PDE4B (0.41) TNKS2CRHR1CRHR2TNKSPDE4B
SCHEMBL20118132 0.90 LMNA (0.46) LMNAESR1TNKS2CRHR1CRHR2
SCHEMBL20118407 0.83 PDE4B (0.40) CRHR1CRHR2PDE4BHTR1A
SCHEMBL20118188 0.82 KDM4E (0.47) TNKS
SCHEMBL20118174 0.82 CRHR1 (0.40) CRHR1CRHR2PDE4BHPGD
SCHEMBL20118184 0.82 CRHR1 (0.39) CRHR1CRHR2PDE4BHPGD
SCHEMBL20103438 0.80 LMNA (0.44) LMNAESR1TNKS2CRHR1CRHR2
SCHEMBL20103162 0.79 LMNA (0.43) LMNAESR1TNKS2CRHR1CRHR2
SCHEMBL20118220 0.77 ALDH1A1 (0.50) CRHR1CRHR2PDE4BHPGD
SCHEMBL20118231 0.77 CRHR1 (0.37) CRHR1CRHR2HPGDHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed