SCHEMBL20135693

SCHEMBL20135693

COCC1(c2ccc(C(=O)OC)c(F)c2)NC(=O)NC1=O

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 1/20 0.42
MMP14 P50281 1/20 0.42
ADAM17 P78536 5/20 0.38
ADAMTS5 Q9UNA0 4/20 0.35
MMP13 P45452 3/20 0.35
MMP2 P08253 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20135529 0.89 MMP14 (0.42) MMP8MMP14ADAM17ADAMTS5MMP13
SCHEMBL20134964 0.81 MMP14 (0.51) MMP8MMP14ADAM17ADAMTS5MMP2
SCHEMBL20135060 0.75 MMP14 (0.45) MMP8MMP14ADAM17ADAMTS5MMP13
SCHEMBL20135676 0.74 MMP8 (0.44) MMP8MMP14ADAM17ADAMTS5MMP13
SCHEMBL20135448 0.73 ADAMTS5 (0.40) ADAM17ADAMTS5MMP13MMP2
SCHEMBL31474027 0.68 CA12 (0.40)
SCHEMBL23163640 0.67 ALDH1A1 (0.41)
SCHEMBL20134812 0.66 MMP14 (0.54) MMP8MMP14ADAM17ADAMTS5MMP13
SCHEMBL20135172 0.66 LMNA (0.52) ADAM17
SCHEMBL5739499 0.65 CA12 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10407408-B2 Imide derivatives and use thereof as medicine MITSUBISHI TANABE PHARMA CORPORATION (JP) 2019-09-10 US disclosed
US-20190077787-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2019-03-14 US disclosed
EP-3321256-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE Mitsubishi Tanabe Pharma Corporation (JP) 2018-05-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190077787-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE MMP9, MMP10, MMP1 MMP8 18/4885MMP14 11/4885ADAM17 36/4885
US-10407408-B2 Imide derivatives and use thereof as medicine MMP9, MMP2, MMP1 MMP8 24/4885MMP14 7/4885ADAM17 39/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.